SCHEMBL30189714

SCHEMBL30189714

CC(C)(C)[Si](C)(C)Oc1cc2ccoc2c([Si](C)(C)C)c1F

nearest known ligand 0.34

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.34
CA12 O43570 4/20 0.31
CA1 P00915 4/20 0.31
CA9 Q16790 4/20 0.31
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
LMNA P02545 1/20 0.30
CYP3A4 P08684 1/20 0.30
HPGD P15428 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
HSD17B10 Q99714 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19783250 1.00 TRPA1 (0.34) TRPA1CA12CA1CA9KDM4E
SCHEMBL28963817 0.77 TRPA1 (0.35) TRPA1KDM4EALDH1A1LMNACYP3A4
SCHEMBL30189920 0.77 CA12 (0.30) CA12CA1CA9
SCHEMBL19782557 0.77 CA12 (0.30) CA12CA1CA9
SCHEMBL29678611 0.74 CA12 (0.33) TRPA1CA12CA1CA9KDM4E
SCHEMBL19783181 0.74 CA12 (0.38) TRPA1CA12CA1CA9KDM4E
SCHEMBL15068207 0.68 CA12 (0.41) CA12CA1CA9CYP3A4
SCHEMBL19782489 0.67 CA12 (0.40) CA12CA1CA9CYP3A4
SCHEMBL15209309 0.63 APLNR (0.38) CA12CA1CA9
SCHEMBL1056366 0.62 ALOX5AP (0.36) TRPA1CA12CA1CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109689647-B Bicyclic heteroaryl substituted compounds 百时美施贵宝公司 2023-01-20 CN disclosed