SCHEMBL30189762

SCHEMBL30189762

COc1cc(C(O)c2cccc(C(F)(F)F)c2)c2nc(Cl)sc2c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
APP P05067 1/20 0.39
ALDH1A1 P00352 2/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
PNMT P11086 1/20 0.38
SCD O00767 1/20 0.36
NR1H4 Q96RI1 1/20 0.36
TAS1R3 Q7RTX0 1/20 0.35
TAS1R1 Q7RTX1 1/20 0.35
TAS1R2 Q8TE23 1/20 0.35
LMNA P02545 1/20 0.35
POLB P06746 1/20 0.35
HTT P42858 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
IDO1 P14902 1/20 0.35
TDO2 P48775 1/20 0.35
CLK1 P49759 1/20 0.35
PPARG P37231 3/20 0.35
GRIN2B Q13224 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19783618 1.00 MEN1 (0.39) MEN1KMT2AAPPALDH1A1L3MBTL1
SCHEMBL19783632 0.88 PNMT (0.41) MEN1KMT2AALDH1A1L3MBTL1PNMT
SCHEMBL30189741 0.88 PNMT (0.41) MEN1KMT2AALDH1A1L3MBTL1PNMT
SCHEMBL21395444 0.79 CYP3A4 (0.39) MEN1KMT2AALDH1A1SCDLMNA
SCHEMBL19783511 0.77 KMT2A (0.38) MEN1KMT2AALDH1A1POLB
SCHEMBL19783775 0.76 F2RL3 (0.55)
SCHEMBL30187628 0.76 F2RL3 (0.55)
SCHEMBL19783627 0.76 ALDH1A1 (0.40) MEN1KMT2AALDH1A1L3MBTL1LMNA
SCHEMBL30189938 0.76 ALDH1A1 (0.40) MEN1KMT2AALDH1A1L3MBTL1LMNA
SCHEMBL19783475 0.74 KMT2A (0.36) KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109689647-B Bicyclic heteroaryl substituted compounds 百时美施贵宝公司 2023-01-20 CN disclosed