SCHEMBL30210345

SCHEMBL30210345

Nc1ccc2nc(-c3ccccn3)cc(N)c2c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.51
TP53 P04637 4/20 0.51
SMN1; SMN2 Q16637 4/20 0.51
L3MBTL1 Q9Y468 4/20 0.51
LMNA P02545 3/20 0.51
NPC1 O15118 2/20 0.51
PKM P14618 2/20 0.51
RAB9A P51151 2/20 0.51
MAPT P10636 2/20 0.51
GAA P10253 1/20 0.51
HPGD P15428 1/20 0.51
METAP2 P50579 1/20 0.51
NPSR1 Q6W5P4 1/20 0.51
ACHE P22303 1/20 0.46
TLR9 Q9NR96 1/20 0.45
METAP1 P53582 4/20 0.45
CCR1 P32246 3/20 0.45
CCR5 P51681 3/20 0.45
CCR8 P51685 3/20 0.45
HSP90AA1 P07900 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30368831 0.85 ACHE (0.64) KDM4ELMNANPSR1ACHEMETAP1
SCHEMBL2712210 0.85 ACHE (0.64) KDM4ELMNANPSR1ACHEMETAP1
SCHEMBL4824379 0.80 ACHE (0.71) KDM4ESMN1; SMN2LMNANPC1PKM
SCHEMBL4244311 0.80 KDM4E (0.47) KDM4ETP53SMN1; SMN2L3MBTL1LMNA
SCHEMBL20652904 0.78 KDM4E (0.56) KDM4ETP53SMN1; SMN2L3MBTL1LMNA
SCHEMBL4251618 0.77 ACHE (0.45) KDM4ETP53SMN1; SMN2L3MBTL1LMNA
SCHEMBL29041842 0.77 ADORA2A (0.52) KDM4ETP53SMN1; SMN2L3MBTL1LMNA
SCHEMBL5048878 0.74 ACHE (0.53) KDM4ELMNANPC1RAB9AMAPT
SCHEMBL4251042 0.74 CCR1 (0.47) KDM4ETP53SMN1; SMN2L3MBTL1LMNA
SCHEMBL4825118 0.74 HSP90AA1 (0.50) KDM4ETP53SMN1; SMN2NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115996939-A AKT3 modulators 乔治穆内有限责任公司 2023-04-21 CN disclosed
CN-115867562-A AKT3 modulators 乔治穆内有限责任公司 2023-03-28 CN disclosed