SCHEMBL30212976

SCHEMBL30212976

COc1cc(N)c(C=O)cc1-c1c(C)cccc1C

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.43
TSHR P16473 2/20 0.43
KDM4E B2RXH2 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
ERN1 O75460 5/20 0.41
TLR2 O60603 1/20 0.41
TLR1 Q15399 1/20 0.41
TLR6 Q9Y2C9 1/20 0.41
DHFR P00374 1/20 0.37
CYP19A1 P11511 1/20 0.37
FFAR1 O14842 1/20 0.37
MAPT P10636 1/20 0.37
PRKDC P78527 1/20 0.37
FGFR1 P11362 1/20 0.36
APP P05067 2/20 0.36
LMNA P02545 1/20 0.36
HPGD P15428 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24027942 1.00 ALDH1A1 (0.43) ALDH1A1TSHRKDM4ETDP1ERN1
SCHEMBL24027895 0.84 ALDH1A1 (0.47) ALDH1A1TSHRKDM4ETDP1ERN1
SCHEMBL12577688 0.84 ERN1 (0.43) ALDH1A1TSHRKDM4ETDP1ERN1
SCHEMBL24027926 0.84 ERN1 (0.47) ALDH1A1TDP1ERN1TLR2TLR1
SCHEMBL30212834 0.84 ALDH1A1 (0.47) ALDH1A1TSHRKDM4ETDP1ERN1
SCHEMBL18359658 0.76 ERN1 (0.55) ERN1
SCHEMBL1570740 0.76 ALDH1A1 (0.72) ALDH1A1TSHRKDM4ETDP1ERN1
SCHEMBL31469616 0.76 ALDH1A1 (0.72) ALDH1A1TSHRKDM4ETDP1ERN1
SCHEMBL27753912 0.76 ALDH1A1 (0.72) ALDH1A1TSHRKDM4ETDP1ERN1
SCHEMBL30011114 0.76 FFAR1 (0.42) ALDH1A1KDM4ETDP1DHFRFFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115697974-A Imidazole 3-oxide derivative based ACSS2 inhibitors and methods of use thereof 美特波米德有限公司 2023-02-03 CN disclosed