SCHEMBL30213802

SCHEMBL30213802

Cc1c([N+](=O)[O-])cnc2c1c(C1=CCN(C(=O)OC(C)(C)C)CC1)cn2C

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PDK4 Q16654 1/20 0.43
BTK Q06187 1/20 0.42
GRM1 Q13255 10/20 0.41
GRM5 P41594 9/20 0.41
SCN9A Q15858 1/20 0.41
EED O75530 2/20 0.41
RBBP4 Q09028 2/20 0.41
SUZ12 Q15022 2/20 0.41
EZH2 Q15910 2/20 0.41
HTR6 P50406 1/20 0.40
GPR119 Q8TDV5 1/20 0.40
CDK9 P50750 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17495396 1.00 PDK4 (0.43) PDK4BTKGRM1GRM5SCN9A
SCHEMBL17963864 0.90 PDK4 (0.42) PDK4BTKGRM1GRM5SCN9A
SCHEMBL17628977 0.89 GRM1 (0.41) PDK4BTKGRM1GRM5SCN9A
SCHEMBL17495445 0.87 POLB (0.33)
SCHEMBL28570087 0.84 NAMPT (0.37)
SCHEMBL17495407 0.84 SCN9A (0.47) PDK4BTKGRM1GRM5SCN9A
SCHEMBL17628762 0.82 P2RX3 (0.34) BTKGRM5GPR119
SCHEMBL17628816 0.82 ALDH1A1 (0.30)
SCHEMBL17629003 0.82
SCHEMBL17495421 0.81 SCN9A (0.47) PDK4GRM1GRM5SCN9AEED

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112759588-B Benzo five-membered heterocyclic amine derivative and application thereof 复旦大学 2023-01-31 CN disclosed