SCHEMBL3021815

SCHEMBL3021815

CCNCc1cccc(-c2ccn3c(-c4cccc(C(=O)NC)c4)cnc3c2)c1

nearest known ligand 0.50

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
KDR P35968 14/20 0.50
FGFR3 P22607 12/20 0.50
FGFR1 P11362 1/20 0.48
FYN P06241 4/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3020569 0.89 KDR (0.51) KDRFGFR3FYN
SCHEMBL13336647 0.81 KDR (0.65) KDRFGFR3FGFR1FYN
Formic Acid SCHEMBL3318748 0.80 KDR (0.61) KDRFGFR3FGFR1FYN
SCHEMBL3030841 0.79 ATM (0.57) KDRFGFR3FGFR1FYN
SCHEMBL27811179 0.79 KDR (0.48) KDRFGFR3FGFR1FYN
SCHEMBL3025894 0.78 KDR (0.50) KDRFGFR3FYN
SCHEMBL3033146 0.78 KDR (0.56) KDRFGFR3FGFR1FYN
SCHEMBL3027808 0.77 FLT3 (0.52) KDRFGFR3
SCHEMBL3029778 0.77 FGFR3 (0.50) KDRFGFR3FGFR1FYN
SCHEMBL3034200 0.77 FGFR3 (0.55) KDRFGFR3FGFR1FYN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101827844-B Imidazo [1,2-a] pyridine derivatives useful as ALK inhibitors NOVARTIS AG 2013-08-14 CN disclosed
US-8367662-B2 Organic compounds NOVARTIS AG (CH) 2013-02-05 US disclosed
EP-2212323-B1 IMIDAZO [1,2-A] PYRIDINE DERIVATIVES USEFUL AS ALK INHIBITORS NOVARTIS AG (CH) 2012-08-15 EP disclosed
CN-101827844-A Imidazo [1,2-a] pyridine derivatives useful as ALK inhibitors NOVARTIS AG 2010-09-08 CN disclosed
US-20100210641-A1 Organic Compounds NOVARTIS AG (CH) 2010-08-19 US disclosed
EP-2212323-A2 IMIDAZO [1,2-A] PYRIDINE DERIVATIVES USEFUL AS ALK INHIBITORS Novartis AG (CH) 2010-08-04 EP disclosed
WO-2009050183-A2 IMIDAZO [1, 2-A] PYRIDINE DERIVATIVES USEFUL AS ALK INHIBITORS NOVARTIS AG (CH) 2009-04-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100210641-A1 Organic Compounds ALK, ACVR1, ACVRL1 KDR 372/4885FGFR3 32/4885FGFR1 72/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.