SCHEMBL30220512

SCHEMBL30220512

CCOC(=O)c1cc2ccnc(OC3CC3)c2n1C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.38
JMJD6 Q6NYC1 2/20 0.38
HCRTR1 O43613 5/20 0.38
HCRTR2 O43614 5/20 0.38
ENPP2 Q13822 1/20 0.38
ALDH1A1 P00352 2/20 0.37
LMNA P02545 1/20 0.37
PIK3CA P42336 1/20 0.37
MAPT P10636 1/20 0.36
HPGD P15428 1/20 0.36
MAPK1 P28482 1/20 0.36
CLK1 P49759 1/20 0.36
UBE2N P61088 1/20 0.36
HSD17B10 Q99714 1/20 0.36
NOS3 P29474 1/20 0.35
NOS1 P29475 1/20 0.35
NOS2 P35228 1/20 0.35
KDM4E B2RXH2 1/20 0.35
CRHBP P24387 1/20 0.35
CRHR2 Q13324 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24896464 0.85 KDM4E (0.39) HCRTR1HCRTR2ALDH1A1HPGDHSD17B10
SCHEMBL30220538 0.82 DHODH (0.40) MAOAJMJD6ALDH1A1LMNAPIK3CA
SCHEMBL30220598 0.80 DGAT1 (0.40) HCRTR1HCRTR2ENPP2ALDH1A1PIK3CA
SCHEMBL30220535 0.79 JMJD6 (0.41) JMJD6ALDH1A1LMNAMAPTMAPK1
SCHEMBL30220530 0.77 SMN1; SMN2 (0.41) JMJD6ALDH1A1PIK3CAMAPTKDM4E
SCHEMBL30220571 0.77 CDC7 (0.41) JMJD6ALDH1A1PIK3CAMAPTHPGD
SCHEMBL25003510 0.77 ACACB (0.35) ACACB
SCHEMBL30220568 0.76 KDM4E (0.45) JMJD6ALDH1A1MAPTHPGDHSD17B10
SCHEMBL24896382 0.76 GRM4 (0.35) ACACB
SCHEMBL24896463 0.74 LRRK2 (0.38) HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4370207-A1 BICYCLIC COMPOUNDS AS ANDROGEN RECEPTOR MODULATORS Nido Biosciences, Inc. (US) 2024-05-22 EP disclosed
WO-2023287704-A1 BICYCLIC COMPOUNDS AS ANDROGEN RECEPTOR MODULATORS NIDO BIOSCIENCES, INC. (US) 2023-01-19 WO disclosed