SCHEMBL30224567

SCHEMBL30224567

[2H]c1ccc2c(cnn2CC(F)(F)F)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RECQL P46063 2/20 0.42
CYP1A2 P05177 2/20 0.40
KMO O15229 1/20 0.39
ADRA2A P08913 1/20 0.35
P2RX7 Q99572 1/20 0.34
DAO P14920 1/20 0.33
PTGS2 P35354 1/20 0.32
POLB P06746 3/20 0.32
CYP17A1 P05093 1/20 0.32
MAPK1 P28482 1/20 0.31
HSD17B10 Q99714 2/20 0.31
NPC1 O15118 2/20 0.31
RAB9A P51151 2/20 0.31
TSHR P16473 2/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
HTR2A P28223 2/20 0.31
HTR2C P28335 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30392789 0.94 RECQL (0.42) RECQLCYP1A2KMOADRA2AP2RX7
SCHEMBL23993150 0.86 RECQL (0.56) RECQLCYP1A2KMOADRA2AP2RX7
SCHEMBL29989569 0.73 CYP17A1 (0.44) RECQLCYP1A2KMOCYP17A1HTR2A
SCHEMBL29355368 0.73 CYP1A2 (0.45) RECQLCYP1A2KMOADRA2AP2RX7
SCHEMBL29353804 0.73 CRHR1 (0.42) RECQLCYP1A2KMOADRA2ANPC1
SCHEMBL29487730 0.71 RECQL (0.46) RECQLCYP1A2KMOADRA2AP2RX7
SCHEMBL25434947 0.71 CYP1A2 (0.36) RECQLCYP1A2CYP17A1HTR2AHTR2C
SCHEMBL30896807 0.71 HTR2A (0.42) KMOADRA2AHTR2AHTR2C
SCHEMBL23994190 0.71 KMO (0.55) CYP1A2KMOADRA2ACYP17A1HTR2A
SCHEMBL24338531 0.71 KMO (0.55) CYP1A2KMOADRA2ACYP17A1HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4143194-A1 CD73 INHIBITING 2,4-DIOXOPYRIMIDINE COMPOUNDS GILEAD SCIENCES, INC. (US) 2023-03-08 EP disclosed