SCHEMBL30228243

SCHEMBL30228243

CCc1nn(C)c(Cc2cccnc2-c2ccc(F)cc2COc2cc(Br)cnc2N)c1Br

nearest known ligand 0.32

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MAP4K3 Q8IVH8 1/20 0.32
MAPK14 Q16539 1/20 0.31
NPC1 O15118 1/20 0.31
HTT P42858 1/20 0.31
RAB9A P51151 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
GRM5 P41594 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28998941 1.00 MAP4K3 (0.32) MAP4K3MAPK14NPC1HTTRAB9A
SCHEMBL30228003 0.85 GRM5 (0.32) MAP4K3NPC1HTTRAB9ASMN1; SMN2
SCHEMBL28998917 0.85 GRM5 (0.32) MAP4K3NPC1HTTRAB9ASMN1; SMN2
SCHEMBL28982110 0.79
SCHEMBL28982112 0.72 JAK2 (0.41)
SCHEMBL30295575 0.72 JAK2 (0.41)
SCHEMBL30242765 0.72 NPC1 (0.34) NPC1RAB9AGRM5
SCHEMBL25624480 0.72 NPC1 (0.34) NPC1RAB9AGRM5
SCHEMBL24014348 0.72 GRM5 (0.32) GRM5
SCHEMBL26537434 0.71 ADCY10 (0.35) MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115916196-A Heteroaromatic macrocyclic ether chemotherapeutic agents 纽威伦特公司 2023-04-04 CN disclosed
EP-4146205-A1 HETEROAROMATIC MACROCYCLIC ETHER CHEMOTHERAPEUTIC AGENTS Nuvalent, Inc. (US) 2023-03-15 EP disclosed