SCHEMBL3024872

SCHEMBL3024872

CC(C)NC(=O)C1CN(C(=O)OCc2ccccc2)CCN1C(=O)OC(C)(C)C

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.54
CTRB1 P17538 1/20 0.48
HTT P42858 1/20 0.48
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
PDK1 Q15118 1/20 0.47
PDK2 Q15119 1/20 0.47
PDK3 Q15120 1/20 0.47
PDK4 Q16654 1/20 0.47
MMP1 P03956 1/20 0.45
MMP3 P08254 1/20 0.45
MMP7 P09237 1/20 0.45
MMP9 P14780 1/20 0.45
MMP13 P45452 1/20 0.45
KMT2A Q03164 3/20 0.45
MEN1 O00255 2/20 0.45
GPR119 Q8TDV5 1/20 0.45
KLK7 P49862 1/20 0.44
CTSL P07711 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5889141 0.96 CTRB1 (0.51) PARP1CTRB1HTTNPC1RAB9A
SCHEMBL9247790 0.88 PARP1 (0.54) PARP1HTTNPC1RAB9ASMN1; SMN2
SCHEMBL7059242 0.87 PARP1 (0.53) PARP1HTTNPC1RAB9ASMN1; SMN2
SCHEMBL1992243 0.87 SMN1; SMN2 (0.62) PARP1HTTNPC1RAB9ASMN1; SMN2
SCHEMBL957813 0.86 PARP1 (0.58) PARP1HTTNPC1RAB9ASMN1; SMN2
SCHEMBL1375861 0.86 PARP1 (0.58) PARP1HTTNPC1RAB9ASMN1; SMN2
SCHEMBL3766378 0.86 PARP1 (0.58) PARP1HTTNPC1RAB9ASMN1; SMN2
SCHEMBL2820733 0.85 PARP1 (0.55) PARP1HTTNPC1RAB9ASMN1; SMN2
SCHEMBL20129643 0.85 PARP1 (0.55) PARP1HTTNPC1RAB9ASMN1; SMN2
SCHEMBL13681760 0.85 PARP1 (0.55) PARP1HTTNPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010178-B1 SUBSTITUTED IMIDAZOLE 4-CARBOXAMIDES AS CHOLECYSTOKININ-1 RECEPTOR MODULATORS MERCK SHARP & DOHME (US) 2010-09-01 EP disclosed