SCHEMBL30252532

SCHEMBL30252532

N#Cc1ccc(-c2nccs2)nc1-c1ccccn1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 2/20 0.48
HSP90AA1 P07900 1/20 0.40
ADORA2A P29274 3/20 0.40
ADORA1 P30542 3/20 0.40
PDPK1 O15530 1/20 0.38
KDM4E B2RXH2 4/20 0.38
ALDH1A1 P00352 3/20 0.38
GAA P10253 2/20 0.38
HPGD P15428 2/20 0.38
HCRTR1 O43613 1/20 0.38
GLA P06280 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
METAP1 P53582 1/20 0.37
SYK P43405 1/20 0.36
SCN9A Q15858 2/20 0.36
CYP19A1 P11511 1/20 0.36
PDE10A Q9Y233 1/20 0.36
MAPT P10636 2/20 0.35
MEN1 O00255 1/20 0.35
USP2 O75604 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20911188 0.77 KDM4E (0.47) RAB9AHSP90AA1ADORA2AADORA1PDPK1
SCHEMBL8936053 0.76 KDM4E (0.47) RAB9AHSP90AA1KDM4EALDH1A1GAA
SCHEMBL452340 0.75 KDM4E (0.57) RAB9AHSP90AA1PDPK1KDM4EALDH1A1
Fluoride SCHEMBL27903468 0.74 KDM4E (0.55) RAB9AHSP90AA1PDPK1KDM4EALDH1A1
Ammonia Solution, Strong SCHEMBL28442530 0.74 KDM4E (0.55) RAB9AHSP90AA1PDPK1KDM4EALDH1A1
SCHEMBL3290082 0.73 PDPK1 (0.43) RAB9AADORA2AADORA1PDPK1KDM4E
SCHEMBL28554182 0.71 KDM4E (0.49) RAB9AHSP90AA1KDM4EALDH1A1GAA
SCHEMBL2651653 0.71 KDM4E (0.48) RAB9AHSP90AA1KDM4EALDH1A1GAA
SCHEMBL29741178 0.71 KDM4E (0.48) RAB9AHSP90AA1KDM4EALDH1A1GAA
SCHEMBL4902877 0.70 RAB9A (0.61) RAB9AHSP90AA1PDPK1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109651358-B 4-aminopyridine derivative, pharmaceutical composition, preparation method and application thereof 上海迪诺医药科技有限公司 2023-04-07 CN disclosed