SCHEMBL30256409

SCHEMBL30256409

CC(C)(C)OC(=O)N1CCc2cccc(OCCCC(=O)OCc3ccccc3)c2[C@H]1CN1C(=O)c2ccccc2C1=O

nearest known ligand 0.43

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.43
PTGDR2 Q9Y5Y4 1/20 0.41
KEAP1 Q14145 12/20 0.40
GHSR Q92847 4/20 0.39
NFE2L2 Q16236 4/20 0.38
ATM Q13315 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
ALDH1A1 P00352 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30258583 1.00 PARP1 (0.43) PARP1PTGDR2KEAP1GHSRNFE2L2
SCHEMBL23930760 0.90 PARP1 (0.45) PARP1PTGDR2KEAP1NFE2L2ATM
SCHEMBL30256353 0.90 KEAP1 (0.44) PARP1PTGDR2KEAP1NFE2L2ATM
SCHEMBL25264776 0.90 KEAP1 (0.44) PARP1PTGDR2KEAP1NFE2L2ATM
SCHEMBL25187459 0.90 KEAP1 (0.44) PARP1PTGDR2KEAP1NFE2L2ATM
SCHEMBL23959356 0.86 KEAP1 (0.41) KEAP1NFE2L2ATML3MBTL1ALDH1A1
SCHEMBL30256146 0.86 KEAP1 (0.41) KEAP1NFE2L2ATML3MBTL1ALDH1A1
SCHEMBL25555241 0.86 KEAP1 (0.41) KEAP1NFE2L2ATML3MBTL1ALDH1A1
SCHEMBL30533745 0.84 KEAP1 (0.44) KEAP1NFE2L2ATML3MBTL1ALDH1A1
SCHEMBL24174323 0.84 KEAP1 (0.41) PARP1KEAP1GHSRNFE2L2ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115667242-B Tetrahydroisoquinoline compounds as NRF2 activators 希四克斯探索有限公司 2025-02-28 CN disclosed
CN-115667242-A Tetrahydroisoquinoline compounds as NRF2 activators 希四克斯探索有限公司 2023-01-31 CN disclosed