SCHEMBL30260968

SCHEMBL30260968

COC(=O)c1ccc2c(-c3nc(Cl)ncc3C(F)(F)F)c[nH]c2c1

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CCNK O75909 15/20 0.51
CDK12 Q9NYV4 15/20 0.51
CCNE1 P24864 9/20 0.51
CDK2 P24941 9/20 0.51
CCNT1 O60563 7/20 0.51
CDK9 P50750 7/20 0.51
CDK7 P50613 6/20 0.50
CCNH P51946 6/20 0.50
MNAT1 P51948 6/20 0.50
EIF2AK2 P19525 1/20 0.47
PDGFRB P09619 1/20 0.46
ASH1L Q9NR48 1/20 0.45
NPC1 O15118 1/20 0.43
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
LMNA P02545 1/20 0.43
HTT P42858 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21178282 1.00 CCNK (0.51) CCNKCDK12CCNE1CDK2CCNT1
SCHEMBL26043639 0.89 CCNK (0.52) CCNKCDK12CCNE1CDK2CCNT1
SCHEMBL26043638 0.88 CCNK (0.51) CCNKCDK12CCNE1CDK2CCNT1
SCHEMBL30261038 0.82 GSK3B (0.47) CCNKCDK12CCNE1CDK2CCNT1
SCHEMBL17683297 0.82 GSK3B (0.47) CCNKCDK12CCNE1CDK2CCNT1
SCHEMBL25363465 0.81 CCNE1 (0.41) CCNKCDK12CCNE1CDK2CCNT1
SCHEMBL31122437 0.81 CCNE1 (0.41) CCNKCDK12CCNE1CDK2CCNT1
SCHEMBL21629046 0.81 CCNK (0.44) CCNKCDK12CCNE1CDK2CCNT1
SCHEMBL30554768 0.81 CCNK (0.44) CCNKCDK12CCNE1CDK2CCNT1
SCHEMBL30957590 0.80 TDO2 (0.47) CCNKCDK12CCNE1CDK2CCNT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250145632-A1 Pyrimidine Heterocyclic Compound, Preparation Method Thereof and use Thereof in Medicine INSILICO MEDICINE IP LIMITED (HK) 2025-05-08 US disclosed
EP-4455132-A1 PYRIMIDINE HETEROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR AND USE THEREOF IN MEDICINE Insilico Medicine IP Limited (HK) 2024-10-30 EP disclosed
CN-118647607-A Pyrimidine heterocyclic compounds, process for preparing the same and pharmaceutical use thereof 英矽智能科技(上海)有限公司 2024-09-13 CN disclosed
EP-4295852-A2 PIPERIDINE DERIVATIVES AS INHIBITORS OF CYCLIN DEPENDENT KINASE 7 (CDK7) Syros Pharmaceuticals, Inc. (US) 2023-12-27 EP disclosed
EP-3484871-B1 PIPERIDINE DERIVATIVES AS INHIBITORS OF CYCLIN DEPENDENT KINASE 7 (CDK7) SYROS PHARMACEUTICALS INC (US) 2023-06-07 EP disclosed
WO-2023040998-A1 A CYCLIN-DEPENDENT KINASE INHIBITOR Taizhou Eoc Pharma Co., Ltd. (CN) 2023-03-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250145632-A1 Pyrimidine Heterocyclic Compound, Preparation Method Thereof and use Thereof in Medicine DPYD, TYMP, NUDT1 CCNK 174/4885CDK12 98/4885CCNE1 315/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.