SCHEMBL30279331

SCHEMBL30279331

COc1cccc(CNC(=O)c2cc(Cl)c(C(=O)O)c(Cl)c2)c1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP13 P45452 3/20 0.68
HPGD P15428 2/20 0.61
LMNA P02545 1/20 0.61
APEX1 P27695 1/20 0.60
RAB9A P51151 1/20 0.59
PRKACA P17612 2/20 0.58
PRKX P51817 2/20 0.58
PRKCQ Q04759 2/20 0.58
ROCK1 Q13464 2/20 0.58
ROCK2 O75116 1/20 0.58
CYP3A4 P08684 1/20 0.58
CYP2D6 P10635 1/20 0.58
CYP2C9 P11712 1/20 0.58
GSK3A P49840 1/20 0.58
GSK3B P49841 1/20 0.58
CLK4 Q9HAZ1 1/20 0.58
ALDH1A1 P00352 3/20 0.57
HTT P42858 1/20 0.57
SMN1; SMN2 Q16637 1/20 0.57
AURKA O14965 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3872357 1.00 MMP13 (0.68) MMP13HPGDLMNAAPEX1RAB9A
SCHEMBL23978716 0.90 MMP13 (0.68) MMP13HPGDLMNAAPEX1RAB9A
SCHEMBL3866898 0.83 MMP13 (0.47) MMP13HPGDLMNAAPEX1RAB9A
SCHEMBL23978699 0.83 NPC1 (0.59) APEX1RAB9ACYP3A4CYP2D6CYP2C9
SCHEMBL6355147 0.83 MMP13 (0.68) MMP13HPGDLMNAAPEX1RAB9A
SCHEMBL7134254 0.83 MMP13 (0.86) MMP13HPGDLMNAAPEX1RAB9A
SCHEMBL30336905 0.82 ROCK2 (0.54) HPGDRAB9AROCK1ROCK2CYP3A4
SCHEMBL3867075 0.82 ROCK2 (0.54) HPGDRAB9AROCK1ROCK2CYP3A4
SCHEMBL28963736 0.82 HPGD (0.60) MMP13HPGDLMNAAPEX1RAB9A
SCHEMBL30112098 0.82 HPGD (0.60) MMP13HPGDLMNAAPEX1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4142707-A1 INHIBITORS OF ALPHA 2 BETA 1 INTEGRIN AND METHODS OF USE THEREOF The Regents of the University of California (US) 2023-03-08 EP disclosed