SCHEMBL30279387

SCHEMBL30279387

COC(=O)[C@H](CNC(=O)N[C@@H]1CCc2ccccc21)NC(=O)OCc1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 4/20 0.53
USP2 O75604 1/20 0.53
TSHR P16473 1/20 0.48
CASP1 P29466 1/20 0.48
HRH1 P35367 1/20 0.48
CTSK P43235 4/20 0.47
ALDH1A1 P00352 2/20 0.46
KYNU Q16719 1/20 0.45
HTT P42858 1/20 0.45
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
ACHE P22303 1/20 0.44
ALOX15 P16050 1/20 0.44
SIRT5 Q9NXA8 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29019148 0.92 EPHX2 (0.55) EPHX2USP2CASP1HRH1CTSK
SCHEMBL30083843 0.87 EPHX2 (0.50) EPHX2USP2CASP1ALDH1A1HTT
SCHEMBL24804772 0.87 EPHX2 (0.50) EPHX2USP2CASP1ALDH1A1HTT
SCHEMBL24805458 0.87 EPHX2 (0.50) EPHX2USP2CASP1ALDH1A1HTT
SCHEMBL24106073 0.85 USP2 (0.54) EPHX2USP2TSHRALDH1A1HTT
SCHEMBL23979138 0.84 USP2 (0.58) EPHX2USP2TSHRALDH1A1HTT
SCHEMBL23978779 0.83 EPHX2 (0.54) EPHX2USP2TSHRALDH1A1HTT
SCHEMBL23978737 0.83 EPHX2 (0.58) EPHX2USP2TSHRALDH1A1HTT
SCHEMBL23978767 0.81 EPHX2 (0.58) EPHX2USP2TSHRALDH1A1HTT
SCHEMBL23978772 0.81 EPHX2 (0.58) EPHX2USP2TSHRALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4142707-A1 INHIBITORS OF ALPHA 2 BETA 1 INTEGRIN AND METHODS OF USE THEREOF The Regents of the University of California (US) 2023-03-08 EP disclosed