SCHEMBL30320627

SCHEMBL30320627

Cn1nc(-c2ccc(N)c(Cl)c2)c2c(N)ncnc21

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 15/20 0.65
PIK3CA P42336 15/20 0.65
PIK3CB P42338 15/20 0.65
PRKDC P78527 15/20 0.65
ABL1 P00519 15/20 0.65
SRC P12931 15/20 0.65
PIK3CG P48736 14/20 0.65
EGFR P00533 14/20 0.65
HCK P08631 14/20 0.65
MTOR P42345 13/20 0.65
EPHB4 P54760 13/20 0.65
KDR P35968 13/20 0.65
PI4KB Q9UBF8 6/20 0.64
NUDT14 O95848 1/20 0.57
NUDT5 Q9UKK9 1/20 0.57
RIPK1 Q13546 1/20 0.51
DAPK3 O43293 1/20 0.50
RIPK2 O43353 1/20 0.50
CYP1A2 P05177 1/20 0.50
LCK P06239 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21436859 1.00 PIK3CD (0.65) PIK3CDPIK3CAPIK3CBPRKDCABL1
SCHEMBL13201532 0.88 PIK3CD (0.70) PIK3CDPIK3CAPIK3CBPRKDCABL1
SCHEMBL23997199 0.85 SRC (0.73) PIK3CDPIK3CAPIK3CBPRKDCABL1
SCHEMBL130598 0.85 SRC (0.75) PIK3CDPIK3CAPIK3CBPRKDCABL1
SCHEMBL130500 0.85 PIK3CA (0.76) PIK3CDPIK3CAPIK3CBPRKDCABL1
SCHEMBL21436578 0.84 PIK3CD (0.65) PIK3CDPIK3CAPIK3CBPRKDCABL1
SCHEMBL30320603 0.84 PIK3CD (0.65) PIK3CDPIK3CAPIK3CBPRKDCABL1
SCHEMBL23917212 0.84 PIK3CD (0.79) PIK3CDPIK3CAPIK3CBPRKDCABL1
SCHEMBL24096629 0.84 SRC (0.84) PIK3CDPIK3CAPIK3CBPRKDCABL1
SCHEMBL30320624 0.84 SRC (0.84) PIK3CDPIK3CAPIK3CBPRKDCABL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112236429-B Heteroaryl compounds useful as type II IRAK inhibitors and uses thereof 默克专利有限公司 2024-10-11 CN disclosed
CN-116075513-A Inhibitors of NEK7 kinase 哈利亚治疗公司 2023-05-05 CN disclosed
EP-4161933-A1 INHIBITORS OF NEK7 KINASE Halia Therapeutics, Inc. (US) 2023-04-12 EP disclosed