SCHEMBL303274

SCHEMBL303274

Nc1cccc2c1CC=NC2

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CD44 P16070 1/20 0.40
ALDH1A1 P00352 2/20 0.35
HPGD P15428 2/20 0.35
KDM4E B2RXH2 2/20 0.35
MAPT P10636 2/20 0.35
MEN1 O00255 1/20 0.35
LMNA P02545 1/20 0.35
GAA P10253 1/20 0.35
KMT2A Q03164 1/20 0.35
TSHR P16473 3/20 0.32
CYP3A4 P08684 3/20 0.32
HSD17B10 Q99714 2/20 0.32
TDP1 Q9NUW8 1/20 0.32
HIF1A Q16665 1/20 0.31
PLAU P00749 1/20 0.31
PIK3CA P42336 1/20 0.31
HTR5A P47898 4/20 0.31
ALOX15 P16050 1/20 0.31
CASP1 P29466 1/20 0.31
CASP7 P55210 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12045032 0.78 HTR5A (0.36) CD44ALDH1A1HPGDPLAUHTR5A
SCHEMBL16111186 0.78 TRPA1 (0.37) PLAU
SCHEMBL586180 0.74 CD44 (0.42) CD44ALDH1A1HPGDKDM4EMAPT
SCHEMBL8527304 0.71 CD44 (0.44) CD44ALDH1A1HPGDKDM4EMAPT
SCHEMBL518391 0.70 PLAU (0.41) TSHRPLAUHTR5A
Hydrochloric Acid SCHEMBL9980683 0.70 CD44 (0.42) CD44ALDH1A1HPGDKDM4EMAPT
SCHEMBL586954 0.69 CD44 (0.47) CD44ALDH1A1HPGDKDM4EMAPT
Hydrochloric Acid SCHEMBL8823227 0.69 PLAU (0.40) TSHRPLAU
SCHEMBL10348095 0.67 CD44 (0.48) CD44ALDH1A1HPGDKDM4EMAPT
SCHEMBL12328333 0.67

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2012500853-A 2012-01-12 JP claimed
EP-2328871-A2 HEDGEHOG PATHWAY MODULATORS IRM LLC (BM) 2011-06-08 EP claimed
WO-2010027746-A2 HEDGEHOG PATHWAY MODULATORS IRM LLC (BM) 2010-03-11 WO claimed
EP-2328871-A2 HEDGEHOG PATHWAY MODULATORS IRM LLC (BM) 2011-06-08 EP disclosed
WO-2010027746-A2 HEDGEHOG PATHWAY MODULATORS IRM LLC (BM) 2010-03-11 WO disclosed