SCHEMBL3033377

SCHEMBL3033377

O=C(c1ccc(Cl)cc1)c1ccc(Br)cn1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.55
ALDH1A1 P00352 1/20 0.55
NPC1 O15118 3/20 0.48
RAB9A P51151 3/20 0.48
CNR2 P34972 1/20 0.47
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
P4HTM Q9NXG6 2/20 0.44
SRD5A2 P31213 1/20 0.44
MAPK1 P28482 1/20 0.44
SMN1; SMN2 Q16637 3/20 0.43
MAPT P10636 2/20 0.43
VNN1 O95497 1/20 0.42
LTC4S Q16873 1/20 0.42
LMNA P02545 1/20 0.42
PRNP P04156 1/20 0.41
HSD17B1 P14061 1/20 0.41
HSD17B2 P37059 1/20 0.41
CES2 O00748 1/20 0.41
CES1 P23141 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27477768 0.90 KDM4E (0.50) KDM4EALDH1A1NPC1RAB9ACNR2
SCHEMBL4603510 0.85 KDM4E (0.53) KDM4EALDH1A1NPC1RAB9AMEN1
SCHEMBL27296576 0.83 KDM4E (0.55) KDM4EALDH1A1NPC1RAB9AMEN1
SCHEMBL13606933 0.83 ALDH1A1 (0.55) KDM4EALDH1A1NPC1RAB9AMEN1
SCHEMBL256768 0.82 ALDH1A1 (0.63) KDM4EALDH1A1NPC1RAB9ACNR2
SCHEMBL5260070 0.79 RAB9A (0.65) KDM4EALDH1A1NPC1RAB9AMEN1
SCHEMBL1267102 0.78 NPC1 (0.66) KDM4EALDH1A1NPC1RAB9AMEN1
SCHEMBL4602074 0.78 ALDH1A1 (0.49) KDM4EALDH1A1NPC1RAB9ASRD5A2
SCHEMBL17157509 0.77 KDM4E (0.56) KDM4EALDH1A1NPC1RAB9AMEN1
SCHEMBL3156716 0.77 MAPK1 (0.64) ALDH1A1RAB9ACNR2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018080065-A1 ORGANIC COMPOUND AND ORGANIC ELECTROLUMINESCENT DEVICE COMPRISING SAME 주식회사 두산 2018-05-03 WO disclosed
US-20100210617-A1 Aryl-Alkylamines And Heteroaryl-Alkylamines As Protein Kinase Inhibitors ASTEX THERAPEUTICS LIMITED (GB) 2010-08-19 US disclosed
US-20100210617-A1 Aryl-Alkylamines And Heteroaryl-Alkylamines As Protein Kinase Inhibitors ASTEX THERAPEUTICS LIMITED (GB) 2010-08-19 US disclosed
US-20100210617-A1 Aryl-Alkylamines And Heteroaryl-Alkylamines As Protein Kinase Inhibitors ASTEX THERAPEUTICS LIMITED (GB) 2010-08-19 US disclosed
EP-1904451-A1 ARYL-ALKYLAMINES AND HETEROARYL-ALKYLAMINES AS PROTEIN KINASE INHIBITORS Astex Therapeutics Limited (GB) 2008-04-02 EP disclosed
WO-2006136830-A1 ARYL-ALKYLAMINES AND HETEROARYL-ALKYLAMINES AS PROTEIN KINASE INHIBITORS ASTEX THERAPEUTICS LIMITED (GB) 2006-12-28 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100210617-A1 Aryl-Alkylamines And Heteroaryl-Alkylamines As Protein Kinase Inhibitors ERBB2, ABL1, GRK2 KDM4E 442/4885ALDH1A1 4220/4885NPC1 3338/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.