SCHEMBL30353060

SCHEMBL30353060

Cn1nc(-c2ccccc2)cc1Oc1cc(C#N)ccc1-c1ncc(CN)cn1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 1/20 0.41
CYP19A1 P11511 2/20 0.40
CYP11B1 P15538 2/20 0.40
CYP11B2 P19099 2/20 0.40
NSD2 O96028 7/20 0.38
PIN1 Q13526 1/20 0.38
PHGDH O43175 1/20 0.36
GRM5 P41594 2/20 0.35
PRKDC P78527 1/20 0.34
PTGDR2 Q9Y5Y4 1/20 0.34
SQOR Q9Y6N5 1/20 0.34
KDM4E B2RXH2 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
RXFP1 Q9HBX9 1/20 0.34
ICMT O60725 1/20 0.33
CYP1A1 P04798 1/20 0.33
CYP1B1 Q16678 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25554317 1.00 SCN9A (0.41) SCN9ACYP19A1CYP11B1CYP11B2NSD2
SCHEMBL25554247 0.93 CYP11B1 (0.41) SCN9ACYP19A1CYP11B1CYP11B2NSD2
SCHEMBL25555418 0.91 CYP19A1 (0.37) SCN9ACYP19A1CYP11B1CYP11B2NSD2
SCHEMBL30353051 0.90 SCN9A (0.40) SCN9ACYP19A1CYP11B1CYP11B2NSD2
SCHEMBL25554271 0.90 SCN9A (0.40) SCN9ACYP19A1CYP11B1CYP11B2NSD2
SCHEMBL25555450 0.89 SCN9A (0.38) SCN9ACYP11B1CYP11B2NSD2
SCHEMBL25057937 0.89 GRM5 (0.37) CYP19A1CYP11B1CYP11B2NSD2GRM5
SCHEMBL30353049 0.89 GRM5 (0.37) CYP19A1CYP11B1CYP11B2NSD2GRM5
SCHEMBL25555451 0.88 NSD2 (0.35) SCN9ACYP19A1CYP11B1CYP11B2NSD2
SCHEMBL25555412 0.88 NSD2 (0.36) SCN9ACYP19A1CYP11B1CYP11B2NSD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115996910-A Aryl or heteroaryl derivatives 帝人制药株式会社 2023-04-21 CN claimed
CN-115996910-A Aryl or heteroaryl derivatives 帝人制药株式会社 2023-04-21 CN disclosed