SCHEMBL30353087

SCHEMBL30353087

Cc1cc(Oc2cc(C#N)ccc2-c2ccc(CCN)cn2)cc(N2CCCC2)n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.42
NPSR1 Q6W5P4 2/20 0.42
ALDH1A1 P00352 2/20 0.42
HTT P42858 2/20 0.42
LMNA P02545 2/20 0.42
POLB P06746 1/20 0.42
AKT1 P31749 2/20 0.34
PIK3CA P42336 2/20 0.34
MTOR P42345 2/20 0.34
GPBAR1 Q8TDU6 2/20 0.33
ERG P11308 1/20 0.33
KDM1A O60341 1/20 0.33
MAPT P10636 1/20 0.33
RECQL P46063 1/20 0.33
HRH4 Q9H3N8 1/20 0.33
CYP11B1 P15538 2/20 0.32
CYP11B2 P19099 2/20 0.32
EGLN2 Q96KS0 1/20 0.32
MEN1 O00255 1/20 0.32
CYP1A2 P05177 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25554212 1.00 TSHR (0.42) TSHRNPSR1ALDH1A1HTTLMNA
SCHEMBL25554066 0.93 PIK3CA (0.42) TSHRNPSR1ALDH1A1HTTLMNA
SCHEMBL30353095 0.93 PIK3CA (0.42) TSHRNPSR1ALDH1A1HTTLMNA
SCHEMBL30353124 0.90 ALDH1A1 (0.41) TSHRNPSR1ALDH1A1HTTLMNA
SCHEMBL25554226 0.90 ALDH1A1 (0.41) TSHRNPSR1ALDH1A1HTTLMNA
SCHEMBL25058564 0.89 CYP19A1 (0.36) TSHRNPSR1ALDH1A1HTTLMNA
SCHEMBL25554594 0.88 SCN7A (0.34) TSHRNPSR1ALDH1A1HTTLMNA
SCHEMBL25554612 0.88 EP300 (0.35) TSHRNPSR1ALDH1A1HTTLMNA
SCHEMBL30353111 0.86 PIK3CA (0.43) TSHRNPSR1ALDH1A1HTTLMNA
SCHEMBL25554350 0.86 PIK3CA (0.43) TSHRNPSR1ALDH1A1HTTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115996910-A Aryl or heteroaryl derivatives 帝人制药株式会社 2023-04-21 CN claimed
CN-115996910-A Aryl or heteroaryl derivatives 帝人制药株式会社 2023-04-21 CN disclosed