SCHEMBL30353151

SCHEMBL30353151

CCOc1cnc(SC)nc1Nc1cc(C)[nH]n1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.43
HTT P42858 1/20 0.43
KMT2A Q03164 1/20 0.43
HSD17B10 Q99714 1/20 0.43
GRM5 P41594 7/20 0.42
AURKA O14965 8/20 0.41
GSK3B P49841 7/20 0.41
AURKB Q96GD4 5/20 0.41
IGF1R P08069 3/20 0.41
SRC P12931 3/20 0.41
FGFR1 P11362 2/20 0.41
KDR P35968 2/20 0.41
INSR P06213 1/20 0.41
PLK4 O00444 1/20 0.40
PAK4 O96013 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30353136 0.82 JAK2 (0.51) MEN1HTTKMT2AHSD17B10AURKA
SCHEMBL30353142 0.80 MEN1 (0.42) MEN1HTTKMT2AHSD17B10GRM5
SCHEMBL28259064 0.73 ALDH1A1 (0.43) MEN1HTTKMT2AGSK3B
SCHEMBL18166030 0.73 IGF1R (0.46) MEN1KMT2AAURKAGSK3BAURKB
SCHEMBL29487435 0.73 IGF1R (0.46) MEN1KMT2AAURKAGSK3BAURKB
SCHEMBL18166072 0.72 PLK4 (0.46) AURKAGSK3BAURKBIGF1RSRC
SCHEMBL19990587 0.72 PLK4 (0.52) AURKAAURKBIGF1RPLK4
SCHEMBL18166052 0.70 PLK4 (0.46) AURKAAURKBIGF1RPLK4PAK4
SCHEMBL174770 0.70 PLK4 (0.48) AURKAGSK3BAURKBSRCPLK4
SCHEMBL30353148 0.69 MEN1 (0.47) MEN1HTTKMT2AHSD17B10AURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11612604-B2 Methods of treating cancer with PLK4 inhibitors LUDWIG INSTITUTE FOR CANCER RESEARCH LTD (CH) 2023-03-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11612604-B2 Methods of treating cancer with PLK4 inhibitors PLK4, PLK2, PLK3 MEN1 3546/4885HTT 3372/4885KMT2A 1059/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.