SCHEMBL30359079

SCHEMBL30359079

COc1cccc(C(=O)N2C3CCC2CNC3)n1

nearest known ligand 0.47

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MGLL Q99685 2/20 0.47
KCNK3 O14649 17/20 0.46
KCNK9 Q9NPC2 17/20 0.46
HTR2A P28223 1/20 0.40
HTR2C P28335 1/20 0.40
HTR2B P41595 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22001648 0.93 KCNK3 (0.45) MGLLKCNK3KCNK9
SCHEMBL30359162 0.89 MGLL (0.43) MGLLKCNK3KCNK9HTR2AHTR2C
SCHEMBL30359034 0.84 MGLL (0.44) MGLLKCNK3KCNK9HTR2AHTR2C
SCHEMBL21904749 0.84 KCNK3 (0.48) MGLLKCNK3KCNK9
SCHEMBL30359027 0.83 KCNK3 (0.49) MGLLKCNK3KCNK9HTR2AHTR2C
SCHEMBL22001486 0.83 KCNK3 (0.49) MGLLKCNK3KCNK9HTR2AHTR2C
SCHEMBL20070578 0.79 MGLL (0.45) MGLLKCNK3KCNK9
SCHEMBL30359104 0.79 KCNK3 (0.47) KCNK3KCNK9
SCHEMBL30358990 0.79 KCNK3 (0.46) MGLLKCNK3KCNK9HTR2AHTR2C
SCHEMBL20587815 0.78 KCNK3 (0.51) MGLLKCNK3KCNK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116057057-A Conjugates of alpha 2-adrenoceptor subtype C (alpha-2C) antagonists and TASK1/3 channel blockers for the treatment of sleep apnea 拜耳公司 2023-05-02 CN disclosed