SCHEMBL30359162

SCHEMBL30359162

COc1cccc(C(=O)N2C3CNCC2CC(=O)C3)n1

nearest known ligand 0.43

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MGLL Q99685 3/20 0.43
KCNK3 O14649 12/20 0.41
KCNK9 Q9NPC2 12/20 0.41
HTR2A P28223 1/20 0.40
HTR2C P28335 1/20 0.40
HTR2B P41595 1/20 0.40
ALOX5 P09917 2/20 0.37
RET P07949 1/20 0.36
DDB1 Q16531 1/20 0.35
CRBN Q96SW2 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30359034 0.92 MGLL (0.44) MGLLKCNK3KCNK9HTR2AHTR2C
SCHEMBL30359079 0.89 MGLL (0.47) MGLLKCNK3KCNK9HTR2AHTR2C
SCHEMBL30359007 0.86 MGLL (0.45) MGLLKCNK3KCNK9HTR2AHTR2C
SCHEMBL30359006 0.84 KCNH2 (0.39) MGLLKCNK3KCNK9HTR2CHTR2B
SCHEMBL22001648 0.82 KCNK3 (0.45) MGLLKCNK3KCNK9
SCHEMBL30359125 0.81 KCNK3 (0.41) KCNK3KCNK9HTR2AHTR2CHTR2B
SCHEMBL30359003 0.80 HTR2A (0.42) KCNK3KCNK9HTR2AHTR2CHTR2B
SCHEMBL30359053 0.79 KCNK3 (0.42) KCNK3KCNK9HTR2AHTR2CHTR2B
SCHEMBL21904749 0.78 KCNK3 (0.48) MGLLKCNK3KCNK9
SCHEMBL20070578 0.76 MGLL (0.45) MGLLKCNK3KCNK9ALOX5RET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116057057-A Conjugates of alpha 2-adrenoceptor subtype C (alpha-2C) antagonists and TASK1/3 channel blockers for the treatment of sleep apnea 拜耳公司 2023-05-02 CN disclosed