SCHEMBL30359124

SCHEMBL30359124

O=C(c1ccncc1)N1CC2CCC1CN2

nearest known ligand 0.53

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 6/20 0.53
CHRNA4 P43681 6/20 0.53
CHRNA3 P32297 5/20 0.53
CHRNB4 P30926 4/20 0.53
CHRNA7 P36544 3/20 0.53
GAA P10253 1/20 0.43
PIK3CD O00329 1/20 0.43
RECQL P46063 2/20 0.43
NPC1 O15118 1/20 0.42
KDM4E B2RXH2 2/20 0.41
KDM1A O60341 1/20 0.39
CHRNB3 Q05901 1/20 0.38
CHRNA6 Q15825 1/20 0.38
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11777276 0.87 CHRNB2 (0.46) CHRNB2CHRNA4CHRNA3CHRNB4CHRNA7
SCHEMBL3335936 0.79 CHRNB2 (0.52) CHRNB2CHRNA4CHRNA3CHRNB4CHRNA7
SCHEMBL3330896 0.79 CHRNB2 (0.52) CHRNB2CHRNA4CHRNA3CHRNB4CHRNA7
SCHEMBL30359051 0.77 HTT (0.51) KDM1A
SCHEMBL30359168 0.74 ALDH1A1 (0.49) KDM4EKDM1A
SCHEMBL31581057 0.74 CCNC (0.54)
SCHEMBL30359139 0.73 PIK3CD (0.47) PIK3CDCYP2C9CYP2C19
SCHEMBL30359097 0.73 MEN1 (0.45) KDM4ECYP2C9CYP2C19
SCHEMBL30359193 0.73 CNR2 (0.43) CHRNB2CHRNA4CHRNA3KDM1ACHRNB3
SCHEMBL3528872 0.73 CHRNB2 (0.53) CHRNB2CHRNA4CHRNA3CHRNB4CHRNA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116057057-A Conjugates of alpha 2-adrenoceptor subtype C (alpha-2C) antagonists and TASK1/3 channel blockers for the treatment of sleep apnea 拜耳公司 2023-05-02 CN disclosed