SCHEMBL30359152

SCHEMBL30359152

O=C(c1ccccc1F)N1C2CNCC1C2

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
ALDH1A1 P00352 3/20 0.44
ALOX15 P16050 1/20 0.44
TSHR P16473 2/20 0.44
KDM4E B2RXH2 3/20 0.44
HTT P42858 3/20 0.43
CES2 O00748 1/20 0.43
CES1 P23141 1/20 0.43
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
MAPK14 Q16539 1/20 0.42
HSD11B1 P28845 2/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
TP53 P04637 1/20 0.41
LMNA P02545 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30359019 0.92 MEN1 (0.50) MEN1KMT2AALDH1A1TSHRKDM4E
SCHEMBL30359059 0.87 MEN1 (0.43) MEN1KMT2AALDH1A1TSHRKDM4E
SCHEMBL20587811 0.84 MEN1 (0.46) MEN1KMT2AALDH1A1TSHRKDM4E
SCHEMBL30359130 0.84 MEN1 (0.46) MEN1KMT2AALDH1A1TSHRKDM4E
SCHEMBL30359107 0.78 MEN1 (0.41) MEN1KMT2AALDH1A1TSHRKDM4E
SCHEMBL20589067 0.78 KCNK3 (0.42) MEN1KMT2AALDH1A1TSHRKDM4E
SCHEMBL30359077 0.75 ALDH1A1 (0.48) KMT2AALDH1A1HTTCYP2C9CYP2C19
SCHEMBL30790488 0.75 SLC6A4 (0.46) ALOX15TSHRLMNA
SCHEMBL30359010 0.73 SLC6A2 (0.46) ALDH1A1LMNA
SCHEMBL10243703 0.73 MEN1 (0.50) MEN1KMT2AALDH1A1KDM4EHSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116057057-A Conjugates of alpha 2-adrenoceptor subtype C (alpha-2C) antagonists and TASK1/3 channel blockers for the treatment of sleep apnea 拜耳公司 2023-05-02 CN disclosed