SCHEMBL30361925

SCHEMBL30361925

Fc1ccc(-c2nn(CCOC(F)F)cc2-c2ncc3cc(-c4ccccc4)oc3n2)cc1

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 1/20 0.37
PTGS2 P35354 2/20 0.35
ABCC1 P33527 7/20 0.33
ABCG2 Q9UNQ0 7/20 0.33
ABCB1 P08183 6/20 0.33
PDE10A Q9Y233 2/20 0.32
FAAH O00519 1/20 0.31
PTGIR P43119 1/20 0.31
ADORA1 P30542 1/20 0.31
EGFR P00533 2/20 0.31
CSNK1D P48730 2/20 0.31
MAP4K4 O95819 1/20 0.31
FRK P42685 1/20 0.31
MAPK9 P45984 1/20 0.31
SLK Q9H2G2 1/20 0.31
CSNK1E P49674 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30362000 0.88 PTGS2 (0.35) S1PR1PTGS2ABCC1ABCG2ABCB1
SCHEMBL30361987 0.87 S1PR1 (0.44) S1PR1PTGS2FAAHADORA1EGFR
SCHEMBL30361895 0.87 PDE10A (0.40) S1PR1PTGS2PDE10A
SCHEMBL30361897 0.87 PTGS2 (0.38) S1PR1PTGS2PDE10AFAAHPTGIR
SCHEMBL30362058 0.85 S1PR1 (0.40) S1PR1PTGS2FAAHADORA1EGFR
SCHEMBL26133085 0.82 EGFR (0.42) PTGS2ABCC1ABCG2ABCB1EGFR
SCHEMBL30362033 0.77 ACVR1 (0.37) S1PR1PTGS2FAAH
SCHEMBL30361899 0.77 ACVR1 (0.37) S1PR1PTGS2FAAH
SCHEMBL30362051 0.77 ACVR1 (0.37) S1PR1PTGS2FAAH
SCHEMBL30361857 0.76 S1PR1 (0.33) S1PR1PTGS2EGFRCSNK1DMAP4K4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023076849-A1 INHIBITORS OF EPIDERMAL GROWTH FACTOR RECEPTOR ORIC PHARMACEUTICALS, INC. (US) 2023-05-04 WO disclosed