SCHEMBL30366353

SCHEMBL30366353

CC(=O)N1c2ccc(-c3ccc(N)cc3)cc2CC[C@@H]1C

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 14/20 0.48
PDK2 Q15119 14/20 0.48
PDK3 Q15120 14/20 0.48
PDK4 Q16654 14/20 0.48
ALDH1A1 P00352 2/20 0.46
HTT P42858 2/20 0.46
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
MAPK1 P28482 1/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
NOTUM Q6P988 1/20 0.43
LMNA P02545 1/20 0.43
TSHR P16473 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26072484 1.00 PDK1 (0.48) PDK1PDK2PDK3PDK4ALDH1A1
SCHEMBL26071711 0.89 PDK1 (0.50) PDK1PDK2PDK3PDK4ALDH1A1
SCHEMBL30366340 0.89 PDK1 (0.50) PDK1PDK2PDK3PDK4ALDH1A1
SCHEMBL26071914 0.87 CYP11B1 (0.47) PDK1PDK2PDK3PDK4ALDH1A1
SCHEMBL30366341 0.87 ALDH1A1 (0.45) PDK1PDK2PDK3PDK4ALDH1A1
SCHEMBL30366739 0.86 HSD17B3 (0.48) PDK1PDK2PDK3PDK4ALDH1A1
SCHEMBL30366745 0.86 HSD17B3 (0.48) PDK1PDK2PDK3PDK4ALDH1A1
SCHEMBL14756238 0.86 HSD17B3 (0.48) PDK1PDK2PDK3PDK4ALDH1A1
SCHEMBL30366544 0.86 HSD17B3 (0.48) PDK1PDK2PDK3PDK4ALDH1A1
SCHEMBL26071930 0.86 HSD17B3 (0.48) PDK1PDK2PDK3PDK4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4165045-A1 DUAL KINASE-BROMODOMAIN INHIBITORS Monash University (AU) 2023-04-19 EP disclosed