SCHEMBL303665

SCHEMBL303665

O=Cc1ccncn1

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29576607 1.00
SCHEMBL27411725 0.98
Hydrochloric Acid SCHEMBL27571277 0.98
Hydrochloric Acid SCHEMBL27665874 0.98 HSP90AA1 (0.41)
Bromide SCHEMBL27776140 0.98
Methylamine SCHEMBL2702693 0.93 HSP90AA1 (0.43)
Trifluoroacetic Acid SCHEMBL28489431 0.83 L3MBTL1 (0.37)
SCHEMBL11865773 0.83 P2RX7 (0.42)
SCHEMBL2818091 0.75
SCHEMBL1013800 0.75

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 981 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113164458-B Monoacylglycerol lipase modulators 詹森药业有限公司 2024-09-13 CN claimed
CN-117466942-A Chiral secondary phosphine oxide compound, chiral quinazolinone/pyrimidinone ring derivative based on chiral secondary phosphine oxide compound and application of chiral quinazolinone/pyrimidinone ring derivative 中山大学 2024-01-30 CN claimed
CN-116457355-A 2-amino-3-carbonyl imidazopyridines and pyrazolopyridines compounds 第一生物治疗股份有限公司 2023-07-18 CN claimed
CN-114764064-A Gold magnetic-mediated fluorescence chemical nasal sensor for rapidly typing pathogenic microorganisms 海南大学 2022-07-19 CN claimed
CN-113214282-B AChE/BACE1/GSK3 beta three-target inhibitor, preparation method thereof and application thereof in resisting Alzheimer disease 中国人民解放军北部战区总医院 2022-03-22 CN claimed
CN-113214282-A AChE/BACE1/GSK3 beta three-target inhibitor, preparation method thereof and application thereof in resisting Alzheimer disease 中国人民解放军北部战区总医院 2021-08-06 CN claimed
CN-113164458-A Monoacylglycerol lipase modulators 詹森药业有限公司 2021-07-23 CN claimed
CN-108003154-B Method for synthesizing paliperidone intermediate by using microchannel reactor 黑龙江鑫创生物科技开发有限公司 2021-03-30 CN claimed
CN-107188898-B Process for preparing thienopyrimidine compounds 霍夫曼-拉罗奇有限公司 2019-12-03 CN claimed
CN-106459092-B Compounds for the treatment of spinal muscular atrophy 豪夫迈·罗氏有限公司 2019-10-15 CN claimed
CN-1247586-C Substituted 2-pyrimidinyl-6, 7,8, 9-tetrahydropyrimido [1, 2-A ] pyrimidin-4-one and 7-pyrimidinyl-2, 3-dihydroimidazo [1, 2-A ] pyrimidin-5 (1H) one derivatives for the treatment of neurodegenerative diseases SANOFI AVENTIS SYNTHELABO (FR) 2006-03-29 CN claimed
EP-1620381-A1 HYDROANTHRACENE BASED COMPOUNDS AS ANTICANCER AGENTS Dabur Research Foundation (IN) 2006-02-01 EP claimed
CN-1714083-A Novel pyrimidine-4,6-dicarboxamides for the selective inhibition of collagenases AVENTIS PHARMA GMBH (DE) 2005-12-28 CN claimed
US-6949557-B2 Hydroanthracene based compounds as anticancer agents DABUR RESEARCH FOUNDATION (IN) 2005-09-27 US claimed
CN-1556810-A Substituted 2-pyrimidinyl-6, 7,8, 9-tetrahydropyrimido [1, 2-A ] pyrimidin-4-one and 7-pyrimidinyl-2, 3-dihydroimidazo [1, 2-A ] pyrimidin-5 (1H) one derivatives for the treatment of neurodegenerative diseases ����ɳŵ��-����������˾ 2004-12-22 CN claimed
WO-2004096742-A1 HYDROANTHRACENE BASED COMPOUNDS AS ANTICANCER AGENTS DABUR RESEARCH FOUNDATION (IN) 2004-11-11 WO claimed
US-20040220197-A1 Hydroanthracene based compounds as anticancer agents DABUR RESEARCH FOUNDATION 2004-11-04 US claimed
CN-1449398-A 2-pyridyl-6, 7,8, 9-tetrahydropyrimido [1, 2-a ] pyrimidin-4-one and 7-pyridyl-2, 3-dihydroimidazo [1, 2-a ] pyrimidin-5 (1H) one derivatives SANOFI SYNTHELABO (FR) 2003-10-15 CN claimed
CN-1049430-C Sulfonamide compound, preparation method and application thereof HOFFMANN LA ROCHE (CH) 2000-02-16 CN claimed
CN-1095375-A Novel sulfonamides HOFFMANN LA ROCHE (CH) 1994-11-23 CN claimed