SCHEMBL30366844

SCHEMBL30366844

Cn1cc(-c2ccc(C(=O)N3CCCC3)c(F)c2)c2c(N)ncc(C#N)c21

nearest known ligand 0.47

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MTOR P42345 15/20 0.47
CYP11B1 P15538 1/20 0.46
CYP11B2 P19099 1/20 0.46
KDM1A O60341 2/20 0.46
ALOX5AP P20292 1/20 0.43
FEN1 P39748 1/20 0.43
LRRK2 Q5S007 1/20 0.42
PIK3CA P42336 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30366524 0.83 MAPK1 (0.46) MTORALOX5APFEN1PIK3CA
SCHEMBL30367019 0.70 ALOX5AP (0.48) ALOX5APFEN1
SCHEMBL30366958 0.70 ALOX5AP (0.43) MTORALOX5APFEN1PIK3CA
SCHEMBL31275471 0.66 MAPK1 (0.47)
SCHEMBL7875295 0.64 MTOR (1.00) MTORPIK3CA
SCHEMBL19243723 0.64 MKNK1 (0.59) MTORPIK3CA
SCHEMBL31264760 0.64 EIF2AK3 (0.50)
SCHEMBL31264739 0.64 EIF2AK3 (0.49)
SCHEMBL4724651 0.63 CPS1 (0.56)
SCHEMBL7876966 0.63 MTOR (1.00) MTORPIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115894481-A Nitrogen-containing heteroaryl compound, preparation method and medical application thereof 江苏恒瑞医药股份有限公司 2023-04-04 CN disclosed