SCHEMBL30366958

SCHEMBL30366958

Cc1cccc(Oc2ccc(-c3cn(C)c4c(C#N)cnc(N)c34)cc2F)n1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5AP P20292 9/20 0.43
FEN1 P39748 9/20 0.43
EIF2AK3 Q9NZJ5 2/20 0.39
RIPK1 Q13546 1/20 0.36
RET P07949 1/20 0.35
KDR P35968 2/20 0.35
PIK3CD O00329 1/20 0.35
ABL1 P00519 1/20 0.35
EGFR P00533 1/20 0.35
HCK P08631 1/20 0.35
SRC P12931 1/20 0.35
PIK3CA P42336 1/20 0.35
PIK3CB P42338 1/20 0.35
MTOR P42345 1/20 0.35
PIK3CG P48736 1/20 0.35
EPHB4 P54760 1/20 0.35
PRKDC P78527 1/20 0.35
GRM2 Q14416 2/20 0.35
TEK Q02763 1/20 0.35
AAK1 Q2M2I8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30367019 0.86 ALOX5AP (0.48) ALOX5APFEN1EIF2AK3GRM2AAK1
SCHEMBL30366806 0.86 TEK (0.43) EIF2AK3RIPK1RETKDRSRC
SCHEMBL30366837 0.78 ALOX5AP (0.36) ALOX5APFEN1EIF2AK3RETKDR
SCHEMBL31213920 0.74 FGFR1 (0.49) EGFRBTK
SCHEMBL28981098 0.73 ALOX5AP (0.38) ALOX5APFEN1GRM2
SCHEMBL30717994 0.71 TRPA1 (0.45) ALOX5APFEN1
SCHEMBL30717977 0.71 TRPA1 (0.45) ALOX5APFEN1
SCHEMBL31264744 0.71 EIF2AK3 (0.47) EIF2AK3RIPK1
SCHEMBL30366844 0.70 MTOR (0.47) ALOX5APFEN1PIK3CAMTOR
SCHEMBL30366769 0.70 KDR (0.35) RETKDRTEK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115894481-A Nitrogen-containing heteroaryl compound, preparation method and medical application thereof 江苏恒瑞医药股份有限公司 2023-04-04 CN disclosed