SCHEMBL30367989

SCHEMBL30367989

Cc1cc(-c2c(Cl)nc(Cl)c3cc(O)ccc23)ccc1F

nearest known ligand 0.40

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 16/20 0.40
ESR2 Q92731 16/20 0.40
ESRRB O95718 1/20 0.38
ESRRA P11474 1/20 0.38
TLR8 Q9NR97 2/20 0.35
PTGS1 P23219 1/20 0.35
PTGS2 P35354 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23887779 1.00 ESR1 (0.40) ESR1ESR2ESRRBESRRATLR8
SCHEMBL25544237 0.86 PTGS2 (0.36) PTGS1PTGS2
SCHEMBL30120996 0.82 KDM4E (0.39) TLR8PTGS2
SCHEMBL23887869 0.82 KDM4E (0.39) TLR8PTGS2
SCHEMBL30121049 0.80 PPARD (0.37)
SCHEMBL23887694 0.80 PPARD (0.37)
SCHEMBL23887781 0.77 ENPP3 (0.41)
SCHEMBL23895771 0.75 GCGR (0.37) ESR1ESR2TLR8PTGS2
SCHEMBL25544512 0.73 GCGR (0.34) PTGS1PTGS2
SCHEMBL23887876 0.71 ESR1 (0.35) ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115697969-A 7-or 8-hydroxy-isoquinoline and 7-or 8-hydroxy-quinoline derivatives as alpha-1 antitrypsin modulators for the treatment of alpha-1 antitrypsin deficiency (AATD) 弗特克斯药品有限公司 2023-02-03 CN disclosed