SCHEMBL30370261

SCHEMBL30370261

Fc1ccc2c(Br)c[nH]c2n1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
AXL P30530 1/20 0.48
MAPK1 P28482 1/20 0.35
ADORA2A P29274 1/20 0.35
ADORA1 P30542 1/20 0.35
CCNT1 O60563 3/20 0.34
CDK9 P50750 3/20 0.34
PIM1 P11309 1/20 0.34
HASPIN Q8TF76 1/20 0.34
CDK2 P24941 2/20 0.33
PRKCI P41743 1/20 0.33
CCNA2 P20248 1/20 0.33
CCNA1 P78396 1/20 0.33
CDK5 Q00535 1/20 0.33
CDK5R1 Q15078 1/20 0.33
EGFR P00533 1/20 0.31
CDC7 O00311 1/20 0.31
CCNE1 P24864 1/20 0.31
DBF4 Q9UBU7 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20576173 1.00 AXL (0.48) AXLMAPK1ADORA2AADORA1CCNT1
SCHEMBL28634050 0.79 AXL (0.52) AXLMAPK1ADORA2AADORA1CCNT1
SCHEMBL21273862 0.76 AXL (0.48) AXLMAPK1ADORA2AADORA1CCNT1
SCHEMBL14635390 0.76 ADORA2A (0.50) AXLADORA2AADORA1
SCHEMBL29605205 0.76 ADORA2A (0.50) AXLADORA2AADORA1
Hydrochloric Acid SCHEMBL22717554 0.74 GSK3B (0.37) ADORA2AADORA1CCNT1CDK9CDK2
SCHEMBL21178475 0.72 AXL (0.44) AXLMAPK1CCNT1CDK9PIM1
SCHEMBL30204138 0.72 AXL (0.44) AXLMAPK1CCNT1CDK9PIM1
Hydrochloric Acid SCHEMBL21546039 0.68 HTR2A (0.50)
SCHEMBL30503527 0.68 CDK5 (0.46) AXLMAPK1ADORA2AADORA1CCNT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4447954-A1 HETEROCYCLIC COMPOUNDS AS 5HT2A BIASED AGONISTS Icahn School of Medicine at Mount Sinai (US) 2024-10-23 EP disclosed
WO-2023114472-A1 HETEROCYCLIC COMPOUNDS AS 5HT2A BIASED AGONISTS ICAHN SCHOOL OF MEDICINE AT MOUNT SINAI (US) 2023-06-22 WO disclosed
CN-108727369-B Influenza virus replication inhibitors and uses thereof 广东东阳光药业有限公司 2023-06-09 CN disclosed