SCHEMBL30375173

SCHEMBL30375173

C#Cc1cncc(N2CCCCC2)c1

nearest known ligand 0.71

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 16/20 0.46
CHRNA4 P43681 15/20 0.46
CHRNA3 P32297 6/20 0.46
CHRNB4 P30926 5/20 0.46
CHRNA1 P02708 4/20 0.44
CHRNG P07510 1/20 0.44
CHRNB1 P11230 1/20 0.44
CHRND Q07001 1/20 0.44
CHRNA2 Q15822 1/20 0.44
CHRNA7 P36544 1/20 0.41
CHKA P35790 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29043100 1.00 CHRNB2 (0.46) CHRNB2CHRNA4CHRNA3CHRNB4CHRNA1
SCHEMBL29108020 0.98 CHRNB2 (0.47) CHRNB2CHRNA4CHRNA3CHRNB4CHRNA1
SCHEMBL30665749 0.98 CHRNB2 (0.47) CHRNB2CHRNA4CHRNA3CHRNB4CHRNA1
SCHEMBL30665748 0.95 CHRNB2 (0.47) CHRNB2CHRNA4CHRNA3CHRNB4CHRNA1
SCHEMBL29108032 0.95 CHRNB2 (0.47) CHRNB2CHRNA4CHRNA3CHRNB4CHRNA1
SCHEMBL1538483 0.84 CHRNB2 (0.62) CHRNB2CHRNA4CHRNA1CHRNA7
SCHEMBL23044774 0.83 CHRNA3 (0.46) CHRNB2CHRNA4CHRNA3CHRNB4CHRNA1
SCHEMBL12396830 0.83 CHRNB2 (0.47) CHRNB2CHRNA4CHRNA3CHRNB4CHRNA1
SCHEMBL3186217 0.83 CHRNB2 (0.58) CHRNB2CHRNA4CHRNA3CHRNB4CHRNA1
SCHEMBL30665759 0.83 CHRNB2 (0.47) CHRNB2CHRNA4CHRNA3CHRNB4CHRNA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116102483-B Substituted pyrrole-2, 5-diketone compound and preparation method and application thereof 中国医学科学院药物研究所 2025-01-17 CN disclosed
CN-117069650-A Alkynyl compound, pharmaceutical composition and application thereof 中国医学科学院药物研究所 2023-11-17 CN disclosed
CN-116102483-A Substituted pyrrole-2, 5-diketone compound and preparation method and application thereof 中国医学科学院药物研究所 2023-05-12 CN disclosed