SCHEMBL30385274

SCHEMBL30385274

CC(C)c1cc(-c2nnc(O)n2-c2ccc(CN3CCCCC3)cc2)c(O)cc1O

nearest known ligand 0.50

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 18/20 0.50
HSP90B1 P14625 3/20 0.50
TRAP1 Q12931 3/20 0.50
HSP90AB1 P08238 7/20 0.48
CYP1A2 P05177 1/20 0.48
CYP2D6 P10635 1/20 0.48
MAPK1 P28482 1/20 0.48
PDK1 Q15118 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22354461 0.91 HSP90AA1 (0.48) HSP90AA1HSP90B1TRAP1HSP90AB1PDK1
SCHEMBL28341024 0.90 HSP90AA1 (0.47) HSP90AA1HSP90B1TRAP1HSP90AB1PDK1
SCHEMBL30368851 0.90 HSP90AA1 (0.47) HSP90AA1HSP90B1TRAP1HSP90AB1PDK1
SCHEMBL5002925 0.90 PDK1 (0.52) HSP90AA1HSP90B1TRAP1HSP90AB1PDK1
SCHEMBL15522473 0.90 HSP90AA1 (0.47) HSP90AA1HSP90B1TRAP1HSP90AB1PDK1
Piperazine SCHEMBL28333614 0.89 HSP90AA1 (0.46) HSP90AA1HSP90B1TRAP1HSP90AB1PDK1
Hydrochloric Acid SCHEMBL29529693 0.89 HSP90AA1 (0.46) HSP90AA1HSP90B1TRAP1HSP90AB1PDK1
Hydrochloric Acid SCHEMBL16569190 0.89 HSP90AA1 (0.46) HSP90AA1HSP90B1TRAP1HSP90AB1PDK1
SCHEMBL30985941 0.88 HRH3 (0.46) HSP90AA1HSP90B1TRAP1HSP90AB1PDK1
SCHEMBL22541228 0.88 HRH3 (0.46) HSP90AA1HSP90B1TRAP1HSP90AB1PDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118139860-A PARP-1 degrading agent and application thereof 西藏海思科制药有限公司 2024-06-04 CN disclosed
WO-2023066363-A1 PARP-1 DEGRADATION AGENT AND USE THEREOF 海思科医药集团股份有限公司 2023-04-27 WO disclosed