SCHEMBL30390481

SCHEMBL30390481

CN(C)c1nc(COCc2ccccc2)cc2ccccc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 4/20 0.43
CYP1A2 P05177 4/20 0.39
CYP2D6 P10635 4/20 0.39
CYP3A4 P08684 3/20 0.39
CYP2C19 P33261 3/20 0.39
CYP2C9 P11712 2/20 0.39
USP2 O75604 2/20 0.39
ALOX15 P16050 2/20 0.39
HSD17B10 Q99714 2/20 0.39
MAPK1 P28482 2/20 0.39
CLK4 Q9HAZ1 2/20 0.39
DHODH Q02127 3/20 0.38
SMN1; SMN2 Q16637 4/20 0.38
HTT P42858 2/20 0.38
STAT3 P40763 1/20 0.38
HSP90AB1 P08238 1/20 0.37
HTR2B P41595 1/20 0.37
GBA1 P04062 1/20 0.37
PDE5A O76074 2/20 0.36
LYPLA1 O75608 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3633944 0.75 HTR2A (0.44) TSHRCYP1A2CYP2D6CYP3A4CYP2C19
SCHEMBL25523802 0.72 KDM4E (0.50) TSHRCYP1A2DHODHSMN1; SMN2HTT
Trimethylammonium SCHEMBL27954231 0.70 TSHR (0.79) TSHRMAPK1LYPLA1LYPLA2ALDH1A1
SCHEMBL21865271 0.70 TSHR (0.58) TSHRCYP1A2CYP2C19HSD17B10MAPK1
SCHEMBL5999845 0.68 MEN1 (0.56) TSHRCYP1A2CYP2D6CYP3A4CYP2C19
SCHEMBL30389997 0.68 MEN1 (0.56) TSHRCYP1A2CYP2D6CYP3A4CYP2C19
SCHEMBL31201809 0.68 SMN1; SMN2 (0.43) TSHRCYP1A2CYP2D6CYP3A4CYP2C19
SCHEMBL4237853 0.68 SMN1; SMN2 (0.43) TSHRCYP1A2CYP2D6CYP3A4CYP2C19
SCHEMBL4271429 0.68 MEN1 (0.46) TSHRCYP1A2CYP2D6CYP3A4CYP2C19
SCHEMBL2472038 0.66 TSHR (0.79) TSHRMAPK1ALDH1A1KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115960046-A Preparation method of 1-amino substituted isoquinoline substances 温州大学 2023-04-14 CN disclosed