SCHEMBL30397185

SCHEMBL30397185

CC(C)(C)OC(=O)N(C(=O)OC(C)(C)C)c1cnc(Br)c(C(F)(F)F)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SOS1 Q07889 1/20 0.37
CACNA1B Q00975 2/20 0.36
CACNA1C Q13936 2/20 0.36
CACNA1G O43497 1/20 0.36
CFTR P13569 4/20 0.35
HDAC1 Q13547 1/20 0.34
HDAC8 Q9BY41 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
BACE1 P56817 2/20 0.33
SSTR4 P31391 1/20 0.33
LMNA P02545 1/20 0.33
POLB P06746 1/20 0.33
NOTUM Q6P988 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
RXRA P19793 1/20 0.31
NR1H2 P55055 1/20 0.31
NR1H3 Q13133 1/20 0.31
USP30 Q70CQ3 1/20 0.31
ASPH Q12797 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25262847 1.00 SOS1 (0.37) SOS1CACNA1BCACNA1CCACNA1GCFTR
SCHEMBL23032506 0.84 MEN1 (0.38) SOS1CACNA1BCACNA1CCACNA1GHDAC1
SCHEMBL23032507 0.82 POLQ (0.38) SOS1CACNA1BCACNA1CCACNA1GHDAC1
SCHEMBL21031816 0.82 CACNA1G (0.35) SOS1CACNA1BCACNA1CCACNA1GHDAC1
SCHEMBL21031817 0.81 CACNA1G (0.34) SOS1CACNA1BCACNA1CCACNA1GHDAC1
SCHEMBL30799546 0.76 SOS1 (0.36) SOS1HDAC1HDAC8HDAC6BACE1
SCHEMBL404990 0.76 BACE1 (0.39) SOS1CACNA1BCACNA1CCACNA1GCFTR
SCHEMBL25256413 0.74 HDAC1 (0.31) CACNA1BCACNA1CCACNA1GHDAC1HDAC8
SCHEMBL31038485 0.74 HDAC1 (0.31) CACNA1BCACNA1CCACNA1GHDAC1HDAC8
SCHEMBL31038421 0.74 CFTR (0.40) CFTRHDAC1HDAC8HDAC6BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118451068-A Tri-fused ring derivative inhibitor, preparation method and application thereof 上海翰森生物医药科技有限公司 2024-08-06 CN disclosed
WO-2023125877-A1 TRICYCLIC DERIVATIVE INHIBITOR, PREPARATION METHOD THEREFOR, AND APPLICATION THEREOF 上海翰森生物医药科技有限公司 2023-07-06 WO disclosed
CN-116171154-A Modulators of cystic fibrosis transmembrane conductance regulator 弗特克斯药品有限公司 2023-05-26 CN disclosed