SCHEMBL30403702

SCHEMBL30403702

c1cncc(-c2cc3n(n2)CCOC3)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 4/20 0.46
CYP2C19 P33261 4/20 0.46
CYP2A6 P11509 3/20 0.46
CYP2E1 P05181 2/20 0.46
CYP2B6 P20813 2/20 0.46
HTT P42858 1/20 0.45
PIK3CA P42336 1/20 0.43
PIK3CB P42338 1/20 0.43
PIK3CG P48736 1/20 0.43
ACVR1 Q04771 3/20 0.42
MEN1 O00255 1/20 0.42
RAB9A P51151 1/20 0.42
KMT2A Q03164 1/20 0.42
ALDH1A1 P00352 1/20 0.41
LMNA P02545 1/20 0.41
GAA P10253 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
CYP3A4 P08684 3/20 0.40
GRM5 P41594 2/20 0.40
CYP11B1 P15538 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22768039 0.84 GRM5 (0.48) HTTRAB9AKMT2AALDH1A1SMN1; SMN2
SCHEMBL30403363 0.82 GRM5 (0.46) PIK3CAPIK3CBPIK3CGGRM5CYP1A2
SCHEMBL30405671 0.76 CYP2A6 (0.41) CYP2C9CYP2C19CYP2A6CYP2E1CYP2B6
SCHEMBL16682846 0.75 PDCD1 (0.55) CYP2C9CYP2C19CYP2A6CYP2E1CYP2B6
SCHEMBL30405703 0.72 CYP2A6 (0.42) CYP2C9CYP2C19CYP2A6CYP2E1CYP2B6
SCHEMBL30405582 0.72 CYP2A6 (0.38) CYP2C9CYP2C19CYP2A6CYP2E1CYP2B6
SCHEMBL20456849 0.70 PIK3CD (0.35) PIK3CAPIK3CBPIK3CGMTOR
SCHEMBL16682671 0.70 KDM4E (0.48) CYP2A6ALDH1A1LMNAGAACYP3A4
SCHEMBL29050010 0.69 GRM5 (0.50) GRM5
SCHEMBL29514224 0.69 GRM5 (0.50) GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116171280-A Casein kinase 1 delta modulators 詹森药业有限公司 2023-05-26 CN claimed