SCHEMBL30405703

SCHEMBL30405703

c1cncc(-c2cc3n(n2)CCCO3)c1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 5/20 0.42
CYP2C9 P11712 3/20 0.42
CYP2E1 P05181 2/20 0.42
CYP2B6 P20813 2/20 0.42
CYP2C19 P33261 2/20 0.42
CYP11B2 P19099 4/20 0.41
CYP11B1 P15538 3/20 0.41
CYP3A4 P08684 3/20 0.40
CYP19A1 P11511 1/20 0.39
HTT P42858 1/20 0.38
PIK3CA P42336 2/20 0.38
PIK3CB P42338 1/20 0.38
PIK3CG P48736 1/20 0.38
ALDH1A1 P00352 2/20 0.38
CYP1A2 P05177 2/20 0.38
USP8 P40818 1/20 0.38
PIM1 P11309 1/20 0.38
FYN P06241 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14844897 0.84 MPO (0.44) HTTALDH1A1
SCHEMBL30405199 0.82 CDC7 (0.46) CYP2C9HTTPIK3CAPIK3CBPIK3CG
SCHEMBL14764810 0.78 LRRK2 (0.33) CYP2A6CYP11B2
SCHEMBL16008737 0.75 MAPK14 (0.47) HTTALDH1A1
SCHEMBL18802950 0.74 GRM5 (0.40) HTTALDH1A1
SCHEMBL30403702 0.72 CYP2C9 (0.46) CYP2A6CYP2C9CYP2E1CYP2B6CYP2C19
SCHEMBL30605064 0.71 MAPK14 (0.43) HTTALDH1A1
SCHEMBL29514377 0.69 GRM5 (0.42)
SCHEMBL29050045 0.69 GRM5 (0.42)
SCHEMBL30305796 0.69 CSNK1E (0.50) CYP11B2HTTPIK3CAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116171280-A Casein kinase 1 delta modulators 詹森药业有限公司 2023-05-26 CN disclosed