SCHEMBL3040463

SCHEMBL3040463

CCOC(=O)Oc1cc(Nc2ccc3c(c2)CC2(C3)C(=O)Nc3ncccc32)ncn1

nearest known ligand 0.48

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ADM2 Q7Z4H4 8/20 0.48
CALCB P10092 7/20 0.47
CALCRL Q16602 12/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3036260 0.90 ADM2 (0.48) ADM2CALCBCALCRL
Hydrochloric Acid SCHEMBL3045318 0.89 ADM2 (0.47) ADM2CALCBCALCRL
SCHEMBL549047 0.88 ADM2 (0.48) ADM2CALCBCALCRL
SCHEMBL3036259 0.81 ADM2 (0.50) ADM2CALCBCALCRL
Hydrochloric Acid SCHEMBL548949 0.81 ADM2 (0.49) ADM2CALCBCALCRL
SCHEMBL3040503 0.79 CALCRL (0.44) CALCRL
SCHEMBL3044880 0.79 CALCRL (0.46) ADM2CALCBCALCRL
SCHEMBL550346 0.78 ADM2 (0.50) ADM2CALCBCALCRL
SCHEMBL17023199 0.78 ADM2 (0.50) ADM2CALCBCALCRL
SCHEMBL3168719 0.77 CALCB (0.47) ADM2CALCBCALCRL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2225227-B1 1',3'-Dihydrospiro[imidazolidin-4,2'-inden]-2,5-diones and 1,3-dihydrospiro[inden-2,3']-pyrroles as CGRP antagonists BOEHRINGER INGELHEIM INT (DE) 2015-08-26 EP disclosed
EP-2251339-A2 COMPOUNDS Boehringer Ingelheim International GmbH (DE) 2010-11-17 EP disclosed