SCHEMBL30405199

SCHEMBL30405199

c1cc(-c2cc3n(n2)CCCO3)ccn1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CDC7 O00311 1/20 0.46
MAPK14 Q16539 1/20 0.45
HDAC1 Q13547 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
GRM5 P41594 1/20 0.38
MPO P05164 2/20 0.36
AR P10275 1/20 0.36
ALDH1A1 P00352 1/20 0.33
THRB P10828 1/20 0.33
HTT P42858 1/20 0.33
CYP2C9 P11712 1/20 0.33
KDR P35968 1/20 0.33
GSK3B P49841 1/20 0.32
PIK3CA P42336 1/20 0.32
PIK3CB P42338 1/20 0.32
PIK3CG P48736 1/20 0.32
DYRK1A Q13627 2/20 0.32
ROCK2 O75116 1/20 0.32
ROCK1 Q13464 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14844897 0.86 MPO (0.44) GRM5MPOALDH1A1HTT
SCHEMBL16008737 0.83 MAPK14 (0.47) MAPK14HDAC1HDAC6MPOAR
SCHEMBL30405703 0.82 CYP2A6 (0.42) ALDH1A1HTTCYP2C9PIK3CAPIK3CB
SCHEMBL30605064 0.79 MAPK14 (0.43) MAPK14HDAC1HDAC6ARALDH1A1
SCHEMBL14764810 0.77 LRRK2 (0.33) HDAC1HDAC6MPO
SCHEMBL18802950 0.76 GRM5 (0.40) GRM5ARALDH1A1HTT
SCHEMBL25272227 0.73 KDM4E (0.41) MAPK14ARALDH1A1THRBHTT
SCHEMBL29514377 0.71 GRM5 (0.42) MAPK14HDAC1HDAC6GRM5THRB
SCHEMBL14844846 0.71 PDE4A (0.38) MAPK14GRM5MPOPIK3CA
SCHEMBL29050045 0.71 GRM5 (0.42) MAPK14HDAC1HDAC6GRM5THRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116171280-A Casein kinase 1 delta modulators 詹森药业有限公司 2023-05-26 CN disclosed