SCHEMBL30409174

SCHEMBL30409174

Oc1ccc2ccccc2c1-c1cc2cc(Br)ccc2[nH]1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 1/20 0.54
IDO1 P14902 5/20 0.44
ESR1 P03372 1/20 0.44
POLB P06746 2/20 0.42
AR P10275 1/20 0.41
HSP90AA1 P07900 1/20 0.41
HSP90AB1 P08238 1/20 0.41
KDM4E B2RXH2 1/20 0.40
MEN1 O00255 1/20 0.40
USP2 O75604 1/20 0.40
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
GAA P10253 1/20 0.40
MAPT P10636 1/20 0.40
HPGD P15428 1/20 0.40
ALOX15 P16050 1/20 0.40
KMT2A Q03164 1/20 0.40
HSD17B10 Q99714 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
CYP2A6 P11509 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19608948 0.85 KDM4E (0.53) CYP19A1ESR1POLBKDM4EMEN1
SCHEMBL30409436 0.85 KDM4E (0.53) CYP19A1ESR1POLBKDM4EMEN1
SCHEMBL30409248 0.83 DAO (0.47) POLBHSP90AA1HSP90AB1KDM4EMEN1
SCHEMBL30410032 0.80 HPN (0.46) ESR1POLBHSP90AA1KDM4EMEN1
SCHEMBL8653093 0.79 POLB (0.53) ESR1POLBHSP90AA1HSP90AB1MEN1
SCHEMBL5620225 0.79 POLB (0.53) ESR1POLBHSP90AA1HSP90AB1MEN1
SCHEMBL17422937 0.75 CYP19A1 (0.71) CYP19A1IDO1ESR1KDM4EMEN1
SCHEMBL11474936 0.75 CYP19A1 (0.61) CYP19A1IDO1ESR1POLBAR
SCHEMBL8964895 0.73 KDM4E (0.60) CYP19A1ESR1POLBKDM4EMEN1
SCHEMBL17422783 0.73 CYP19A1 (0.71) CYP19A1IDO1ESR1CYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116102562-B Naphtho [2,1-b ] indolo [2,3-d ] cyclooctalactone derivative and preparation method thereof 江苏师范大学 2024-11-26 CN claimed
CN-116102562-A Naphtho [2,1-b ] indolo [2,3-d ] cyclooctalactone derivative and preparation method thereof 江苏师范大学 2023-05-12 CN claimed
CN-116102562-B Naphtho [2,1-b ] indolo [2,3-d ] cyclooctalactone derivative and preparation method thereof 江苏师范大学 2024-11-26 CN disclosed
CN-116102562-A Naphtho [2,1-b ] indolo [2,3-d ] cyclooctalactone derivative and preparation method thereof 江苏师范大学 2023-05-12 CN disclosed