SCHEMBL30427243

SCHEMBL30427243

N#Cc1cnn(-c2ncccc2Cl)c1

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 1/20 0.45
GRM5 P41594 5/20 0.40
RPS6KA5 O75582 1/20 0.36
DRD2 P14416 2/20 0.36
HTR2A P28223 2/20 0.36
EGLN2 Q96KS0 1/20 0.35
HTR1A P08908 1/20 0.34
HTR7 P34969 1/20 0.34
CYP17A1 P05093 1/20 0.34
CYP1A2 P05177 1/20 0.34
SMO Q99835 1/20 0.34
KDM4D Q6B0I6 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3265565 0.80 PLAU (0.38) CYP17A1CYP1A2
SCHEMBL18394388 0.78 CYP17A1 (0.35) CYP17A1CYP1A2
SCHEMBL950266 0.78 ALDH1A1 (0.44) RPS6KA5CYP17A1CYP1A2
SCHEMBL12528560 0.78 HSD11B1 (0.42) PDE10ACYP17A1CYP1A2
SCHEMBL27686519 0.78 BCHE (0.41) PDE10AGRM5DRD2CYP1A2
SCHEMBL25208515 0.76 EGLN2 (0.35) PDE10AGRM5EGLN2
SCHEMBL29818491 0.76 EGLN2 (0.35) PDE10AGRM5EGLN2
SCHEMBL10910898 0.74 GRM5 (0.66) PDE10AGRM5DRD2
SCHEMBL2559023 0.72 GRM5 (0.34) GRM5
SCHEMBL13484047 0.72 ADORA2A (0.37) GRM5RPS6KA5DRD2HTR2AHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022164789-A9 TRICYCLIC COMPOUNDS USEFUL IN THE TREATMENT OF CANCER, AUTOIMMUNE AND INFLAMMATORY DISORDERS SCHRÖDINGER, INC. (US) 2023-05-25 WO disclosed