SCHEMBL30428263

SCHEMBL30428263

c1ccc(CC2NCC23CCOC3)cc1

nearest known ligand 0.38

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 2/20 0.35
POLB P06746 1/20 0.34
SLC6A2 P23975 1/20 0.34
SLC6A4 P31645 1/20 0.34
SLC6A3 Q01959 1/20 0.34
GBA1 P04062 1/20 0.33
DDB1 Q16531 1/20 0.32
CRBN Q96SW2 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL34463931 0.79 POLB (0.42) HDAC8POLBGBA1DDB1CRBN
SCHEMBL16616098 0.76 GBA1 (0.47) HDAC8POLBGBA1
SCHEMBL31633626 0.73 GBA1 (0.38) HDAC8POLBGBA1
SCHEMBL22227942 0.70 CYP1A2 (0.35)
SCHEMBL30428125 0.65 POLB (0.41) HDAC8POLBGBA1
SCHEMBL17959206 0.64 POLB (0.44) HDAC8POLBGBA1
SCHEMBL28293435 0.63 MAOA (0.45) POLB
SCHEMBL28588930 0.62 GBA1 (0.42) HDAC8POLBSLC6A2SLC6A3GBA1
SCHEMBL23477959 0.62 POLB (0.46) HDAC8POLBGBA1
SCHEMBL23477826 0.62 POLB (0.42) HDAC8POLBGBA1DDB1CRBN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4456895-A2 HETEROARYL COMPOUNDS AS INHIBITORS OF IRAK4, COMPOSITIONS AND APPLICATIONS THEREOF Accro Bioscience (HK) Limited (HK) 2024-11-06 EP disclosed
WO-2023130054-A2 HETEROARYL COMPOUNDS AS INHIBITORS OF IRAK4, COMPOSITIONS AND APPLICATIONS THEREOF ACCRO BIOSCIENCE (HK) LIMITED (CN) 2023-07-06 WO disclosed