SCHEMBL30430258

SCHEMBL30430258

COC(=O)c1c(C)cc(Cl)nc1Cl

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.50
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
MAPK1 P28482 1/20 0.50
CYP3A4 P08684 2/20 0.49
ACHE P22303 1/20 0.49
TAAR1 Q96RJ0 1/20 0.48
HPGD P15428 2/20 0.46
KDM4E B2RXH2 4/20 0.44
POLB P06746 3/20 0.44
HSD17B10 Q99714 2/20 0.44
CASP1 P29466 1/20 0.44
PLA2G2A P14555 1/20 0.40
GLA P06280 1/20 0.40
TSHR P16473 1/20 0.40
NPSR1 Q6W5P4 1/20 0.39
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1085042 1.00 ALDH1A1 (0.50) ALDH1A1MEN1KMT2ASMN1; SMN2MAPK1
SCHEMBL25151051 0.87 CYP3A4 (0.47) ALDH1A1MEN1KMT2ASMN1; SMN2MAPK1
SCHEMBL18786786 0.86 CYP3A4 (0.46) ALDH1A1MEN1KMT2ASMN1; SMN2MAPK1
SCHEMBL24773237 0.86 CYP3A4 (0.50) ALDH1A1MEN1KMT2ASMN1; SMN2MAPK1
SCHEMBL22689984 0.85 ALDH1A1 (0.65) ALDH1A1MEN1KMT2ASMN1; SMN2MAPK1
SCHEMBL1710208 0.85 KDM4E (0.44) ALDH1A1MEN1KMT2ASMN1; SMN2MAPK1
SCHEMBL1085064 0.84 POLB (0.47) ALDH1A1MEN1KMT2ASMN1; SMN2MAPK1
SCHEMBL25343847 0.84 KDM4E (0.54) ALDH1A1MEN1KMT2ASMN1; SMN2MAPK1
SCHEMBL24175026 0.84 CYP3A4 (0.51) ALDH1A1MEN1KMT2ASMN1; SMN2MAPK1
SCHEMBL14660349 0.82 ALDH1A1 (0.43) ALDH1A1MEN1KMT2ASMN1; SMN2MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116134022-B ATR inhibitors and uses thereof 上海德琪医药科技有限公司 2025-03-18 CN disclosed
CN-119212988-A Kinesin KIF18A inhibitor and application thereof 上海湃隆生物科技有限公司 2024-12-27 CN disclosed
CN-116554151-B Kinesin KIF18A inhibitor and application thereof 上海湃隆生物科技有限公司 2024-09-20 CN disclosed
CN-116554151-A Kinesin KIF18A inhibitor and application thereof 上海湃隆生物科技有限公司 2023-08-08 CN disclosed
EP-4175948-A1 ATR INHIBITORS AND USES THEREOF ANTENGENE DISCOVERY LIMITED (CN) 2023-05-10 EP disclosed