SCHEMBL3043079

SCHEMBL3043079

NC(=O)[C@H]1CN(c2ccc3c(c2)OCCc2cn[nH]c2-3)C(=O)O1

nearest known ligand 0.45

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MAOA P21397 2/20 0.45
PIK3CA P42336 8/20 0.37
HSP90AA1 P07900 1/20 0.36
CALML3 P27482 1/20 0.35
KMT2A Q03164 2/20 0.34
GRK2 P25098 1/20 0.34
CTDSP1 Q9GZU7 1/20 0.34
SIGMAR1 Q99720 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3048133 0.90 MAOA (0.36) MAOAPIK3CAHSP90AA1KMT2ASIGMAR1
SCHEMBL3042217 0.89 MAOA (0.36) MAOAPIK3CACALML3SIGMAR1
SCHEMBL6241199 0.87 MAOA (0.43) MAOAHSP90AA1CALML3
SCHEMBL3041022 0.87 MAOA (0.43) MAOAHSP90AA1CALML3
SCHEMBL3042246 0.82 MAOA (0.47) MAOAPIK3CACALML3KMT2AGRK2
SCHEMBL6238879 0.82 MAOA (0.51) MAOACALML3
SCHEMBL6241235 0.82 MAOA (0.51) MAOACALML3
SCHEMBL3045561 0.79 MAOA (0.41) MAOAPIK3CACALML3KMT2AGRK2
SCHEMBL3035586 0.79 MAOA (0.41) MAOAPIK3CAKMT2ASIGMAR1
SCHEMBL3042185 0.79 MAOA (0.41) MAOAPIK3CAKMT2AGRK2CTDSP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040147760-A1 N-aryl-2-oxazolidinone-5-carboxamides and their derivatives PHARMACIA & UPJOHN COMPANY 2004-07-29 US claimed
US-7645781-B2 N-aryl-2-oxazolidinone-5-carboxamides and their derivatives PFIZER INC (US) 2010-01-12 US disclosed
US-7645781-B2 N-aryl-2-oxazolidinone-5-carboxamides and their derivatives PFIZER INC (US) 2010-01-12 US disclosed
US-7645781-B2 N-aryl-2-oxazolidinone-5-carboxamides and their derivatives PFIZER INC (US) 2010-01-12 US disclosed
US-20070015801-A1 N-aryl-2-oxazolidinone-5-carboxamides and their derivatives THOMAS RICHARD C 2007-01-18 US disclosed
US-20070015801-A1 N-aryl-2-oxazolidinone-5-carboxamides and their derivatives THOMAS RICHARD C 2007-01-18 US disclosed
US-20070015801-A1 N-aryl-2-oxazolidinone-5-carboxamides and their derivatives THOMAS RICHARD C 2007-01-18 US disclosed
US-7141588-B2 N-aryl-2-oxazolidinone-5-carboxamides and their derivatives PFIZER, INC. (US) 2006-11-28 US disclosed
US-20040147760-A1 N-aryl-2-oxazolidinone-5-carboxamides and their derivatives PHARMACIA & UPJOHN COMPANY 2004-07-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040147760-A1 N-aryl-2-oxazolidinone-5-carboxamides and their derivatives OXA1L, AADAC, MT-ND5 MAOA 957/4885PIK3CA 2855/4885HSP90AA1 2681/4885
US-20070015801-A1 N-aryl-2-oxazolidinone-5-carboxamides and their derivatives OXA1L, AADAC, MT-ND5 MAOA 957/4885PIK3CA 2855/4885HSP90AA1 2681/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.