SCHEMBL30438361

SCHEMBL30438361

CNCCC(Oc1cccc(C(=O)Nc2cccnc2)c1)c1cccs1

nearest known ligand 0.59

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CACNA2D1 P54289 15/20 0.59
ALDH1A1 P00352 2/20 0.56
TSHR P16473 1/20 0.54
MAPK1 P28482 1/20 0.54
MEN1 O00255 1/20 0.52
NPC1 O15118 1/20 0.52
RAB9A P51151 1/20 0.52
KMT2A Q03164 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
BRAF P15056 1/20 0.52
SLC6A2 P23975 5/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20917067 1.00 CACNA2D1 (0.59) CACNA2D1ALDH1A1TSHRMAPK1MEN1
SCHEMBL22714212 0.89 CACNA2D1 (0.60) CACNA2D1NPC1RAB9AKMT2ASMN1; SMN2
SCHEMBL20917054 0.85 ALDH1A1 (0.60) CACNA2D1ALDH1A1TSHRMAPK1MEN1
SCHEMBL30438714 0.85 ALDH1A1 (0.60) CACNA2D1ALDH1A1TSHRMAPK1MEN1
SCHEMBL20917283 0.85 CACNA2D1 (0.58) CACNA2D1MAPK1MEN1NPC1RAB9A
SCHEMBL20599777 0.81 CACNA2D1 (0.67) CACNA2D1SLC6A2
SCHEMBL20917078 0.81 CACNA2D1 (0.50) CACNA2D1ALDH1A1TSHRMAPK1MEN1
SCHEMBL20917081 0.80 CACNA2D1 (0.57) CACNA2D1SLC6A2
SCHEMBL30438709 0.80 CACNA2D1 (0.57) CACNA2D1SLC6A2
SCHEMBL20917049 0.78 CACNA2D1 (0.57) CACNA2D1SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111225901-B Propylamine derivatives for the treatment of pain and pain-related disorders 埃斯特韦制药股份公司 2023-07-04 CN claimed
CN-111225901-B Propylamine derivatives for the treatment of pain and pain-related disorders 埃斯特韦制药股份公司 2023-07-04 CN disclosed