SCHEMBL30445113

SCHEMBL30445113

Cc1cc(-n2ncc(CO)n2)ncc1C#N

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KCNJ1 P48048 17/20 0.48
KCNH2 Q12809 2/20 0.44
ABCB11 O95342 1/20 0.43
POU2F2 P09086 1/20 0.43
POU2F1 P14859 1/20 0.43
SLC47A1 Q96FL8 1/20 0.43
P2RX7 Q99572 1/20 0.40
KDM4E B2RXH2 1/20 0.34
NPC1 O15118 1/20 0.34
ALDH1A1 P00352 1/20 0.34
RAB9A P51151 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
RXFP1 Q9HBX9 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
MALT1 Q9UDY8 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20168335 1.00 KCNJ1 (0.48) KCNJ1KCNH2ABCB11POU2F2POU2F1
SCHEMBL21243688 0.90 KCNJ1 (0.47) KCNJ1KCNH2ABCB11POU2F2POU2F1
SCHEMBL24135397 0.88 KCNJ1 (0.47) KCNJ1KCNH2ABCB11POU2F2POU2F1
SCHEMBL26536810 0.83 KCNJ1 (0.47) KCNJ1P2RX7KDM4E
SCHEMBL20176738 0.81 KCNJ1 (0.41) KCNJ1KCNH2ABCB11POU2F2POU2F1
SCHEMBL30445215 0.80 KCNJ1 (0.41) KCNJ1KCNH2ABCB11POU2F2POU2F1
SCHEMBL20574336 0.80 KCNJ1 (0.41) KCNJ1KCNH2ABCB11POU2F2POU2F1
SCHEMBL23586685 0.78 KCNJ1 (0.57) KCNJ1KCNH2ABCB11POU2F2POU2F1
SCHEMBL30444639 0.78 KCNJ1 (0.52) KCNJ1KCNH2ABCB11POU2F2POU2F1
SCHEMBL20168367 0.78 KCNJ1 (0.52) KCNJ1KCNH2ABCB11POU2F2POU2F1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110139862-B Substituted bicyclic heterocyclic derivatives useful as ROMK channel inhibitors 百时美施贵宝公司 2024-01-16 CN disclosed
CN-110678463-B Substituted nitrogen-containing compounds 百时美施贵宝公司 2023-06-06 CN disclosed