SCHEMBL30449285

SCHEMBL30449285

C1=Cc2c(cnc3ccccc23)OC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.39
GPR3 P46089 1/20 0.39
CYP2B6 P20813 2/20 0.38
CYP1A2 P05177 8/20 0.35
CYP1A1 P04798 6/20 0.35
CYP1B1 Q16678 6/20 0.35
ERN1 O75460 1/20 0.33
ALDH1A1 P00352 2/20 0.32
GLA P06280 1/20 0.32
GAA P10253 1/20 0.32
HPGD P15428 1/20 0.32
HSD17B10 Q99714 1/20 0.32
NCF1 P14598 1/20 0.31
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31
PI4KA P42356 1/20 0.31
PI4K2B Q8TCG2 1/20 0.31
PI4K2A Q9BTU6 1/20 0.31
PI4KB Q9UBF8 1/20 0.31
PDE4A P27815 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30003732 0.79 MAPT (0.47) KDM4ECYP2B6CYP1A2CYP1A1CYP1B1
SCHEMBL5902340 0.73 KDM4E (0.39) KDM4EGPR3CYP2B6CYP1A2CYP1A1
SCHEMBL30079979 0.71 KDM4E (0.40) KDM4EGPR3ERN1ALDH1A1GLA
SCHEMBL28412569 0.71 CYP1A2 (0.37) CYP2B6CYP1A2CYP1A1CYP1B1ALDH1A1
SCHEMBL28551604 0.70 GPR3 (0.42) KDM4EGPR3ERN1ALDH1A1GLA
SCHEMBL29756136 0.70 CA12 (0.47) KDM4ECYP2B6CYP1A2CYP1A1CYP1B1
SCHEMBL87841 0.70 CA12 (0.47) KDM4ECYP2B6CYP1A2CYP1A1CYP1B1
SCHEMBL1041972 0.70 CA12 (0.47) KDM4ECYP2B6CYP1A2CYP1A1CYP1B1
SCHEMBL29749295 0.70 GPR3 (0.42) KDM4EGPR3ERN1ALDH1A1GLA
SCHEMBL6671643 0.68 CYP1A2 (0.48) CYP2B6CYP1A2CYP1A1CYP1B1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116332948-A Nitrogen-containing tetracyclic compound, preparation method and medicinal application thereof 翰森生物有限责任公司 2023-06-27 CN disclosed