SCHEMBL30449307

SCHEMBL30449307

Cc1cn(-c2cc(F)cc(Cl)c2)c2c1C(O)C(F)(F)CC2

nearest known ligand 0.45

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
EPAS1 Q99814 11/20 0.45
ARNT P27540 7/20 0.45
FFAR4 Q5NUL3 1/20 0.34
VEGFA P15692 5/20 0.33
METAP2 P50579 4/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24109436 1.00 EPAS1 (0.45) EPAS1ARNTFFAR4VEGFAMETAP2
SCHEMBL25800592 0.91 EPAS1 (0.40) EPAS1ARNTVEGFA
SCHEMBL24110079 0.88 EPAS1 (0.44) EPAS1ARNTFFAR4VEGFAMETAP2
SCHEMBL24110056 0.86 EPAS1 (0.43) EPAS1ARNTFFAR4VEGFA
SCHEMBL30449323 0.86 EPAS1 (0.43) EPAS1ARNTFFAR4VEGFA
SCHEMBL24110081 0.85 EPAS1 (0.53) EPAS1ARNTVEGFA
SCHEMBL28980671 0.85 EPAS1 (0.53) EPAS1ARNTVEGFA
SCHEMBL29116096 0.85 EPAS1 (0.53) EPAS1ARNTVEGFA
SCHEMBL25800760 0.85 ALDH1A1 (0.35) EPAS1ARNT
SCHEMBL30449352 0.84 EPAS1 (0.42) EPAS1ARNTFFAR4VEGFA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115884966-B Bicyclic compounds and uses thereof 贝达药业股份有限公司 2024-10-22 CN claimed
CN-115884966-A Bicyclic compounds and uses thereof 贝达药业股份有限公司 2023-03-31 CN claimed
CN-119431335-A Bicyclic compounds and uses thereof 贝达药业股份有限公司 2025-02-14 CN disclosed
CN-115884966-B Bicyclic compounds and uses thereof 贝达药业股份有限公司 2024-10-22 CN disclosed
CN-117126097-A Bicyclic compounds and uses thereof 贝达药业股份有限公司 2023-11-28 CN disclosed
CN-115884966-A Bicyclic compounds and uses thereof 贝达药业股份有限公司 2023-03-31 CN disclosed