SCHEMBL30450157

SCHEMBL30450157

COc1ccc(-c2ccnc(Cl)n2)c(OC)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A1 P04798 4/20 0.52
CYP1B1 Q16678 4/20 0.52
CRHR1 P34998 1/20 0.50
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
NPC1 O15118 3/20 0.46
RAB9A P51151 3/20 0.46
MAPT P10636 2/20 0.46
NFKB1 P19838 2/20 0.46
NFKB2 Q00653 2/20 0.46
RELA Q04206 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
TLR9 Q9NR96 2/20 0.46
ATM Q13315 1/20 0.46
CYP1A2 P05177 1/20 0.45
CYP2E1 P05181 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2C8 P10632 1/20 0.45
CYP2D6 P10635 1/20 0.45
CYP2A6 P11509 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL444455 1.00 CYP1A1 (0.52) CYP1A1CYP1B1CRHR1MEN1KMT2A
SCHEMBL30451078 0.84 CYP1A1 (0.55) CYP1A1CYP1B1CRHR1MEN1KMT2A
SCHEMBL31011620 0.84 HSP90AA1 (0.45) CRHR1MAPTTLR9TSHRGAA
SCHEMBL31011585 0.84 CCNT1 (0.40) CYP1A1CYP1B1CRHR1MEN1KMT2A
SCHEMBL31011609 0.84 HSP90AA1 (0.45) CRHR1MAPTTLR9TSHRGAA
SCHEMBL25339277 0.83 HSP90AA1 (0.55) CYP1A1CYP1B1CYP1A2CYP2E1CYP3A4
SCHEMBL31119002 0.83 HSP90AA1 (0.55) CYP1A1CYP1B1CYP1A2CYP2E1CYP3A4
SCHEMBL31011660 0.82 PDGFRB (0.41) MEN1KMT2ANPC1RAB9AMAPT
SCHEMBL28512792 0.82 GSK3B (0.60) CYP1A1CYP1B1CRHR1MEN1KMT2A
SCHEMBL30507464 0.82 GSK3B (0.60) CYP1A1CYP1B1CRHR1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116253687-A Diaryl pyrimidine compound and preparation method and application thereof 复旦大学 2023-06-13 CN disclosed